SCHEMBL8828342

SCHEMBL8828342

CCCc1ccccc1N1CCN(CCCN)CC1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.55
KDM4E B2RXH2 1/20 0.52
LMNA P02545 1/20 0.52
DRD2 P14416 6/20 0.52
DRD3 P35462 4/20 0.52
HTR1A P08908 3/20 0.52
DRD4 P21917 1/20 0.52
HTR2A P28223 1/20 0.52
HTR2C P28335 1/20 0.52
SIGMAR1 Q99720 2/20 0.51
BRD4 O60885 1/20 0.51
BRD9 Q9H8M2 1/20 0.51
NCF1 P14598 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828449 0.90 DRD2 (0.59) CYP2D6KDM4ELMNADRD2DRD3
SCHEMBL27466797 0.85 CYP2D6 (0.61) CYP2D6KDM4ELMNADRD2DRD3
SCHEMBL6991590 0.82 CYP2D6 (0.58) CYP2D6KDM4ELMNADRD2DRD3
SCHEMBL8828376 0.80 SIGMAR1 (0.59) CYP2D6DRD2DRD3HTR1ADRD4
SCHEMBL13061367 0.80 NCF1 (0.59) LMNADRD2DRD3HTR1ADRD4
SCHEMBL8828565 0.79 CYP2D6 (0.61) CYP2D6DRD2DRD3HTR1AHTR2A
SCHEMBL1541501 0.79 NCF1 (0.63) CYP2D6LMNADRD2DRD3HTR1A
SCHEMBL9559725 0.77 KDM4E (0.68) CYP2D6KDM4ELMNADRD2DRD3
SCHEMBL8828353 0.77 CYP2D6 (0.63) CYP2D6KDM4ELMNADRD2DRD3
SCHEMBL7972648 0.77 CYP2D6 (0.63) CYP2D6KDM4ELMNASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688795-A URINARY TRACTS OBSTRUCTION SYNTEX (U.S.A.) INC. (US) 1997-11-18 US disclosed
EP-0711757-A1 3-(4-phenylpiperazin-1-yl)propyl-amino, thio and oxy -pyridine, pyrimidine and benzene derivatives as alpha1-adrenoceptor antagonists F. Hoffmann-La Roche AG (CH) 1996-05-15 EP disclosed