SCHEMBL8828486

SCHEMBL8828486

O=C(O)c1cnncc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
TSHR P16473 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TP53 P04637 1/20 0.41
CASP1 P29466 1/20 0.41
AKR1C4 P17516 1/20 0.40
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
AKR1C1 Q04828 1/20 0.40
LMNA P02545 1/20 0.39
HCAR2 Q8TDS4 2/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
HAVCR2 Q8TDQ0 1/20 0.37
DAO P14920 1/20 0.37
ALOX15 P16050 1/20 0.36
CYP1A2 P05177 1/20 0.36
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
NAPRT Q6XQN6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL70537 0.81 HCAR2 (0.46) ALDH1A1TSHRSMN1; SMN2LMNAHCAR2
SCHEMBL3523197 0.72 ALDH1A1 (0.42) ALDH1A1TSHRSMN1; SMN2CASP1HCAR2
SCHEMBL5120215 0.70 KMT2A (0.54) ALDH1A1HCAR2KEAP1ALOX15CYP1A2
SCHEMBL353823 0.70 GABRP (0.50) ALDH1A1HCAR2ALOX15CYP1A2KDM4E
SCHEMBL29952809 0.70 GABRP (0.50) ALDH1A1HCAR2ALOX15CYP1A2KDM4E
SCHEMBL29952027 0.70 KMT2A (0.54) ALDH1A1HCAR2KEAP1ALOX15CYP1A2
SCHEMBL29446081 0.70 SMN1; SMN2 (0.47) ALDH1A1TSHRSMN1; SMN2TP53CASP1
SCHEMBL29574646 0.70 ROCK2 (0.58) ALDH1A1TSHRSMN1; SMN2TP53CASP1
SCHEMBL625580 0.70 SMN1; SMN2 (0.47) ALDH1A1TSHRSMN1; SMN2TP53CASP1
SCHEMBL7533 0.70 ROCK2 (0.58) ALDH1A1TSHRSMN1; SMN2TP53CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688795-A URINARY TRACTS OBSTRUCTION SYNTEX (U.S.A.) INC. (US) 1997-11-18 US disclosed
CN-1136039-A [3- (4-phenylpiperazin-1-yl) propylamino, thio and oxy ] -pyridine, pyrimidine and benzene derivatives HOFFMANN LA ROCHE (CH) 1996-11-20 CN disclosed
EP-0711757-A1 3-(4-phenylpiperazin-1-yl)propyl-amino, thio and oxy -pyridine, pyrimidine and benzene derivatives as alpha1-adrenoceptor antagonists F. Hoffmann-La Roche AG (CH) 1996-05-15 EP disclosed