SCHEMBL8828488

SCHEMBL8828488

COc1cc(OCc2ccccc2)ccc1N1CCNCC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.64
SLC6A2 P23975 3/20 0.64
SLC6A4 P31645 3/20 0.64
SLC6A3 Q01959 3/20 0.64
HTR6 P50406 2/20 0.57
HTR3A P46098 3/20 0.56
HTR3E A5X5Y0 2/20 0.56
HTR3B O95264 2/20 0.56
HTR3D Q70Z44 2/20 0.56
HTR3C Q8WXA8 2/20 0.56
ADRB1 P08588 1/20 0.56
DRD2 P14416 1/20 0.56
CYP2C19 P33261 1/20 0.56
DRD3 P35462 1/20 0.56
SIGMAR1 Q99720 1/20 0.56
LMNA P02545 1/20 0.55
MAPT P10636 1/20 0.55
TLR7 Q9NYK1 3/20 0.50
TLR9 Q9NR96 2/20 0.50
NTRK1 P04629 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17658996 0.83 HTR1A (0.72) HTR1ASLC6A2SLC6A4SLC6A3HTR6
SCHEMBL8226269 0.82 HTR1A (0.59) HTR1ASLC6A2SLC6A4SLC6A3HTR6
SCHEMBL7240022 0.82 SLC6A2 (0.55) HTR1ASLC6A2SLC6A4CYP2C19SIGMAR1
Hydrochloric Acid SCHEMBL23783250 0.81 SLC6A2 (0.58) HTR1ASLC6A2SLC6A4SLC6A3HTR6
Hydrochloric Acid SCHEMBL30032096 0.81 SLC6A2 (0.58) HTR1ASLC6A2SLC6A4SLC6A3HTR6
SCHEMBL30747759 0.81 HTR3A (0.71) HTR1AHTR6HTR3AHTR3EHTR3B
SCHEMBL233151 0.81 HTR3A (0.71) HTR1AHTR6HTR3AHTR3EHTR3B
SCHEMBL8257048 0.81 HTR3A (0.52) HTR1ASLC6A2SLC6A4HTR6HTR3A
Hydrochloric Acid SCHEMBL4905371 0.80 HTR3A (0.69) HTR1AHTR6HTR3AHTR3EHTR3B
Hydrochloric Acid SCHEMBL7711668 0.80 HTR3A (0.69) HTR1AHTR6HTR3AHTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688795-A URINARY TRACTS OBSTRUCTION SYNTEX (U.S.A.) INC. (US) 1997-11-18 US disclosed
CN-1136039-A [3- (4-phenylpiperazin-1-yl) propylamino, thio and oxy ] -pyridine, pyrimidine and benzene derivatives HOFFMANN LA ROCHE (CH) 1996-11-20 CN disclosed
EP-0711757-A1 3-(4-phenylpiperazin-1-yl)propyl-amino, thio and oxy -pyridine, pyrimidine and benzene derivatives as alpha1-adrenoceptor antagonists F. Hoffmann-La Roche AG (CH) 1996-05-15 EP disclosed