SCHEMBL8828762

SCHEMBL8828762

CCN(CC)C(=O)c1cnc(NCCCN2CCN(c3ccccc3OC)CC2)nc1

nearest known ligand 0.67

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.58
HTR1A P08908 4/20 0.56
HTR2A P28223 3/20 0.56
HTR7 P34969 3/20 0.56
HTR6 P50406 3/20 0.56
DRD3 P35462 2/20 0.56
DRD4 P21917 1/20 0.56
ADRA1D P25100 1/20 0.56
ADRA1A P35348 1/20 0.56
ADRA1B P35368 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8828753 0.82 ADRA1D (0.58) DRD2DRD3ADRA1DADRA1AADRA1B
SCHEMBL8828767 0.82 ADRA1D (0.73) ADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL9027560 0.81 ADRA1D (0.72) ADRA1DADRA1AADRA1B
SCHEMBL8828464 0.81 DRD2 (0.57) DRD2HTR2A
SCHEMBL9760092 0.75 HTR1A (0.62) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL8828771 0.75 DRD2 (0.54) DRD2HTR7
SCHEMBL9760272 0.75 DRD2 (0.67) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL9027734 0.74 ADRA1D (0.75) ADRA1DADRA1AADRA1B
SCHEMBL9760177 0.74 HTR1A (0.73) DRD2HTR1AHTR2AHTR7HTR6
SCHEMBL9027618 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688795-A URINARY TRACTS OBSTRUCTION SYNTEX (U.S.A.) INC. (US) 1997-11-18 US disclosed
EP-0711757-A1 3-(4-phenylpiperazin-1-yl)propyl-amino, thio and oxy -pyridine, pyrimidine and benzene derivatives as alpha1-adrenoceptor antagonists F. Hoffmann-La Roche AG (CH) 1996-05-15 EP disclosed