SCHEMBL8829977

SCHEMBL8829977

COc1ccc(CNC(=S)CCc2ccco2)c(OC)c1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.68
TAS1R1 Q7RTX1 1/20 0.68
HPGD P15428 5/20 0.56
NPSR1 Q6W5P4 1/20 0.56
POLB P06746 2/20 0.51
ALDH1A1 P00352 7/20 0.47
SMN1; SMN2 Q16637 5/20 0.47
APLNR P35414 1/20 0.47
MAPT P10636 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MEN1 O00255 1/20 0.45
LMNA P02545 1/20 0.45
GAA P10253 1/20 0.45
MAPK1 P28482 1/20 0.45
KMT2A Q03164 1/20 0.45
TDP1 Q9NUW8 2/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL701170 0.81 TAS1R3 (1.00) TAS1R3TAS1R1HPGDNPSR1POLB
SCHEMBL22501325 0.80 TAS1R3 (0.71) TAS1R3TAS1R1HPGDNPSR1POLB
SCHEMBL14817128 0.78 TAS1R3 (0.76) TAS1R3TAS1R1HPGDNPSR1POLB
SCHEMBL4739573 0.75 APLNR (0.56) TAS1R3TAS1R1NPSR1ALDH1A1SMN1; SMN2
SCHEMBL8829967 0.75 TAS1R3 (0.67) TAS1R3TAS1R1HPGDNPSR1POLB
SCHEMBL31016553 0.75 TAS1R3 (0.64) TAS1R3TAS1R1HPGDNPSR1POLB
SCHEMBL13693769 0.74 KMT2A (0.62) NPSR1POLBALDH1A1SMN1; SMN2MAPT
SCHEMBL26324037 0.73 APLNR (0.65) TAS1R3TAS1R1HPGDNPSR1POLB
SCHEMBL4786270 0.72 KMT2A (0.60) POLBALDH1A1SMN1; SMN2APLNRMAPT
SCHEMBL2226834 0.72 APLNR (0.63) TAS1R3TAS1R1HPGDNPSR1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5616711-A REACTING BUTENE DERIVATIVE TO AN AMIDE DERIVATIVE; USEFUL AS INTERMEDIATES FOR PRODUCING ANTIULCER DRUGS FUJIREBIO INC. (JP) 1997-04-01 US disclosed
EP-0582304-A2 Methods of producing amino butene derivatives FUJIREBIO Inc. (JP) 1994-02-09 EP disclosed