SCHEMBL8834058

SCHEMBL8834058

COc1cc(Nc2cc(C(=O)O)c(C(=O)O)cc2Nc2ccccc2)cc(OC)c1OC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.56
AKR1C2 P52895 1/20 0.56
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
BRAF P15056 1/20 0.53
IDO1 P14902 2/20 0.52
TDO2 P48775 2/20 0.52
KDM4E B2RXH2 2/20 0.50
MAPK9 P45984 1/20 0.50
MAPK10 P53779 1/20 0.50
HTT P42858 1/20 0.50
ALDH1A1 P00352 1/20 0.50
HPGD P15428 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
HSD17B10 Q99714 1/20 0.50
RCE1 Q9Y256 1/20 0.50
PTK2 Q05397 3/20 0.49
CTSV O60911 1/20 0.49
CTSL P07711 1/20 0.49
ATM Q13315 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8834423 0.90 MAPT (0.57) AKR1C3AKR1C2MEN1KMT2ABRAF
SCHEMBL8834430 0.89 KDM4E (0.50) AKR1C3AKR1C2MEN1KMT2ABRAF
SCHEMBL5841124 0.81 BRAF (0.69) MEN1KMT2ABRAFATMGAK
SCHEMBL8833788 0.81 MAPT (0.67) AKR1C3AKR1C2MEN1KMT2AKDM4E
SCHEMBL8834506 0.80 AKR1C3 (0.67) AKR1C3AKR1C2MEN1KMT2AKDM4E
SCHEMBL20745310 0.79 KDM4E (0.71) AKR1C3AKR1C2MEN1KMT2AKDM4E
SCHEMBL12072039 0.78 PTK2 (0.73) KDM4EMAPK9MAPK10HTTALDH1A1
SCHEMBL11644754 0.78 AKR1C3 (0.68) AKR1C3AKR1C2KMT2AKDM4EALDH1A1
SCHEMBL27972004 0.78 CTSV (0.58) AKR1C3AKR1C2MEN1KMT2ABRAF
SCHEMBL8833806 0.78 EGFR (0.69) MEN1KMT2ABRAFIDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5663336-A IMIDATION OF DIAMINOPHTHALIC ACID TO FORM KINASE INHIBITORS AS ANTITUMOR AGENTS CIBA-GEIGY CORPORATION (US) 1997-09-02 US disclosed
US-5491144-A KINASE INHIBITORS, ANTITUMOR AGENTS CIBA-GEIGY CORPORATION (US) 1996-02-13 US disclosed