SCHEMBL8835508

SCHEMBL8835508

CC(C)(C)c1c(C(F)(F)F)ccc(C(=O)C(O)c2ccccc2)c1N

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.40
CES2 O00748 3/20 0.40
CES1 P23141 2/20 0.40
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPK1 P28482 1/20 0.36
HPGD P15428 1/20 0.34
HDAC4 P56524 4/20 0.34
HDAC6 Q9UBN7 3/20 0.34
HDAC3 O15379 3/20 0.34
HDAC1 Q13547 3/20 0.34
AOC3 Q16853 1/20 0.33
GAA P10253 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
ACP3 P15309 1/20 0.33
SLC7A5 Q01650 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8835492 0.78 LMNA (0.38) LMNACES2CES1KDM4EALDH1A1
SCHEMBL8542240 0.76 CES2 (0.35) LMNACES2KDM4EALDH1A1MAPK1
SCHEMBL680608 0.74 LMNA (0.52) LMNACES2CES1KDM4EALDH1A1
SCHEMBL28264518 0.72 LMNA (0.46) LMNACES2CES1KDM4EALDH1A1
SCHEMBL9817968 0.72 LMNA (0.46) LMNACES2CES1KDM4EALDH1A1
SCHEMBL545347 0.71 LMNA (0.52) LMNACES2CES1KDM4EALDH1A1
SCHEMBL28956589 0.69 CES2 (0.50) LMNACES2CES1KDM4EALDH1A1
SCHEMBL3516962 0.69 LMNA (0.49) LMNACES2CES1KDM4EALDH1A1
SCHEMBL8671236 0.68 LMNA (0.41) LMNACES2CES1KDM4EALDH1A1
SCHEMBL1476486 0.68 CES2 (0.52) LMNACES2CES1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5703107-A CENTRAL NERVOUS SYSTEM DISORDERS; ANALGESICS; ANTIEPILEPTIC AGENTS MERRELL PHARMACEUTICALS INC. (US) 1997-12-30 US disclosed