SCHEMBL8845652

SCHEMBL8845652

COc1ccc(C(=C2CCCCC2)c2ccc(OC)cc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.64
PGR P06401 1/20 0.64
CHRM2 P08172 1/20 0.64
ADORA3 P0DMS8 1/20 0.64
AR P10275 1/20 0.64
CHRM1 P11229 1/20 0.64
SLC6A2 P23975 1/20 0.64
SLC6A3 Q01959 1/20 0.64
ESR2 Q92731 2/20 0.53
PSMB1 P20618 2/20 0.51
PSMB5 P28074 2/20 0.51
PSMB2 P49721 2/20 0.51
OPRM1 P35372 1/20 0.49
OPRD1 P41143 1/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
HPGD P15428 2/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.49
DPP7 Q9UHL4 2/20 0.47
CES2 O00748 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3468131 0.87 ESR1 (0.51) ESR1PGRCHRM2ADORA3AR
SCHEMBL16265352 0.87 ALDH1A1 (0.54) ESR1PGRCHRM2ADORA3AR
SCHEMBL9256713 0.82 OPRM1 (0.48) ESR1PGRCHRM2ADORA3AR
SCHEMBL19699727 0.82 ESR1 (0.55) ESR1PGRCHRM2ADORA3AR
SCHEMBL8316134 0.81 OPRD1 (0.69) ESR1PGRCHRM2ADORA3AR
Cyclofenil SCHEMBL21045976 0.79 ESR1 (0.94) ESR1PGRCHRM2ADORA3AR
Cyclofenil SCHEMBL132246 0.78 ESR1 (1.00) ESR1PGRCHRM2ADORA3AR
Cyclofenil SCHEMBL11222765 0.78 ESR1 (1.00) ESR1PGRCHRM2ADORA3AR
Cyclofenil SCHEMBL6340459 0.77 ESR1 (0.97) ESR1PGRCHRM2ADORA3AR
SCHEMBL4612699 0.77 NPSR1 (0.50) ESR1PGRCHRM2ADORA3AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5663207-A ADMINISTERING TO INHIBIT DEVELOPMENT OF BREAST TUMOR RESEARCH CORPORATION TECHNOLOGIES (US) 1997-09-02 US disclosed
US-5658914-A ANTIESTROGENS, ANTITUMOR AGENTS RESEARCH CORPORATION TECHNOLOGIES (US) 1997-08-19 US disclosed
US-5658951-A ANTIESTROGENS, ANTITUMOR AGENTS RESEARCH CORPORATION TECHNOLOGIES (US) 1997-08-19 US disclosed
US-5658927-A ANTIESTROGENS, ANTITUMOR AGENTS RESEARCH CORPORATION TECHNOLOGIES (US) 1997-08-19 US disclosed
US-5397802-A Gem-dichlorocyclopropanes as antitumor agents RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1995-03-14 US disclosed
US-4879315-A Cyclopropyl analogs as anti-estrogenic, anti-tumor and female fertility agents THE BOARD OF REGENTS FOR THE UNIVERSITY OF OKLAHOMA (US) 1989-11-07 US disclosed