SCHEMBL8845756

SCHEMBL8845756

CNC(=O)Oc1cc2c(cc1F)N(CCCCc1ccccn1)CC2

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 9/20 0.39
HTR2B P41595 9/20 0.39
HTR2A P28223 7/20 0.39
ALDH1A1 P00352 3/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
HTT P42858 1/20 0.38
HCRTR2 O43614 1/20 0.36
NAAA Q02083 1/20 0.35
GLS O94925 1/20 0.35
HTR1A P08908 1/20 0.34
ADRA1A P35348 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8846262 0.84 ACHE (0.43) HTR2CHTR2BHTR2AALDH1A1L3MBTL1
SCHEMBL8845748 0.84 DRD4 (0.36) HTR2CHTR2BHCRTR2
SCHEMBL8845546 0.66 ITGB3 (0.48) ALDH1A1
SCHEMBL8845742 0.66 TP53 (0.35) HTR2CHTR2BHTR2AHCRTR2
SCHEMBL30376197 0.65 PARP10 (0.43) ALDH1A1L3MBTL1KDM4E
SCHEMBL29374038 0.63 ALDH1A1 (0.62) ALDH1A1L3MBTL1KDM4E
SCHEMBL6636318 0.62 HRH1 (0.43) ALDH1A1L3MBTL1
SCHEMBL6638799 0.62 HRH1 (0.43) ALDH1A1L3MBTL1
SCHEMBL8282497 0.61 NPC1 (0.57) ALDH1A1NAAA
SCHEMBL6801884 0.60 ROCK1 (0.47) ALDH1A1L3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688816-A COGNITION ACTIVATOR; ALZHEIMER'S DISEASE HOECHST MARION ROUSSEL, INC. (US) 1997-11-18 US disclosed
US-5455245-A Alzheimer*s disease HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1995-10-03 US disclosed
US-5264442-A For treating alzheimer's disease HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-11-23 US disclosed
EP-0471298-A1 Carbamoyl-1-(pyridinylalkyl)-1H-indoles, indolines and related analogs HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-02-19 EP disclosed