SCHEMBL8848428

SCHEMBL8848428

O=C(Cl)C1(c2ccc3c(c2)CCCC3)CCC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
HDAC4 P56524 4/20 0.39
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HSD11B1 P28845 1/20 0.36
CFTR P13569 1/20 0.36
LMNA P02545 1/20 0.36
IDO1 P14902 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
KDM4E B2RXH2 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
HPGD P15428 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8847829 0.84 AKR1C1 (0.52) ALDH1A1ALOX15TSHRHSD17B10MEN1
SCHEMBL8848204 0.79 L3MBTL1 (0.45) ALDH1A1HDAC4ALOX15TSHRHSD17B10
SCHEMBL1465052 0.75 ALDH1A1 (0.52) ALDH1A1MEN1KMT2AHPGD
SCHEMBL13551754 0.75 ESR1 (0.33) ALDH1A1HSD11B1
SCHEMBL8105060 0.75 HDAC1 (0.50) SLC6A2SLC6A4
SCHEMBL3443425 0.74 HDAC4 (0.61) ALDH1A1HDAC4HSD11B1LMNAKMT2A
SCHEMBL15800503 0.73 CTNNB1 (0.39) LMNA
SCHEMBL8097178 0.73 HDAC1 (0.47) ALDH1A1HDAC4HSD11B1HPGD
SCHEMBL29275065 0.73 HSD11B1 (0.47) ALDH1A1HDAC4HSD11B1LMNAIDO1
SCHEMBL248544 0.72 AKR1C1 (0.64) ALDH1A1HDAC4HSD11B1LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5663416-A ENZYME INHIBITORS AS ANTIINFLAMMATORY AGENTS OR DERMATITIS TREATMENT CORTECH INC. 1997-09-02 US disclosed
EP-0465802-A1 Oxidant sensitive and insensitive aromatic esters as inhibitors of human neutrophil elastase CORTECH, INC. (US) 1992-01-15 EP disclosed