SCHEMBL8855199

SCHEMBL8855199

COc1cc(C(C)C)c(OC)c2c1C1(C)CCCC(C)(CO)C1CC2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLA1 P09884 2/20 0.51
CYP3A4 P08684 5/20 0.49
ALOX15 P16050 3/20 0.49
MAPT P10636 2/20 0.49
USP2 O75604 1/20 0.49
HPGD P15428 1/20 0.49
TSHR P16473 3/20 0.48
CYP2C9 P11712 2/20 0.48
CYP2C19 P33261 2/20 0.48
KARS1 Q15046 1/20 0.47
FDPS P14324 2/20 0.41
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
MAPK1 P28482 2/20 0.36
PDK1 Q15118 1/20 0.36
PDK2 Q15119 1/20 0.36
PDK3 Q15120 1/20 0.36
PDK4 Q16654 1/20 0.36
CYP2D6 P10635 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8855332 0.82 CYP3A4 (0.54) POLA1CYP3A4ALOX15MAPTUSP2
SCHEMBL9355660 0.71 CYP3A4 (0.33) CYP3A4MAPTUSP2HPGDCYP2C9
SCHEMBL29552651 0.71 FDPS (0.37) CYP3A4ALOX15MAPTUSP2HPGD
SCHEMBL9360485 0.71 LPAR1 (0.33) CYP3A4MAPTUSP2HPGDCYP2C9
SCHEMBL9364236 0.70 CYP3A4 (0.72) POLA1CYP3A4ALOX15MAPTUSP2
SCHEMBL8855272 0.70 MAPT (0.37) CYP3A4MAPTALDH1A1LMNACYP19A1
SCHEMBL8855173 0.70 CYP3A4 (0.31) CYP3A4MAPTALDH1A1
SCHEMBL8855310 0.70 CYP3A4 (0.33) CYP3A4MAPTALDH1A1PIK3CAPIK3CG
18-Hydroxyferruginol SCHEMBL32666150 0.68 KARS1 (0.67) POLA1CYP3A4ALOX15MAPTUSP2
18-Hydroxyferruginol SCHEMBL18290210 0.68 KARS1 (0.67) POLA1CYP3A4ALOX15MAPTUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5654343-A NITRIC OXIDE SYNTHESIS INHIBITOR; TREATING ENDOTOXIC SHOCK OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-08-05 US disclosed
EP-0676196-A1 NITROGEN MONOXIDE SYNTHESIS INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-10-11 EP disclosed