SCHEMBL8856091

SCHEMBL8856091

CCCCCCCCC(CCCCCC)C(=S)Nc1c(Sc2nc[nH]n2)ccc2ncccc12

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ALOX5 P09917 5/20 0.33
PTGES O14684 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
CACNA2D1 P54289 2/20 0.31
HTT P42858 1/20 0.31
TLR8 Q9NR97 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8856179 0.85 TRPV1 (0.36) ALDH1A1SMN1; SMN2ALOX5PTGESTRPV1
SCHEMBL8856352 0.83 TRPV1 (0.35) ALDH1A1SMN1; SMN2ALOX5PTGESTRPV1
SCHEMBL9431040 0.82 ALOX5 (0.37) ALDH1A1SMN1; SMN2ALOX5PTGESTRPV1
SCHEMBL8856361 0.80 TRPV1 (0.37) ALDH1A1SMN1; SMN2ALOX5TRPV1PPARG
SCHEMBL8856078 0.80 ALDH1A1 (0.36) ALDH1A1SMN1; SMN2ALOX5TRPV1PPARG
SCHEMBL8856302 0.79 KMT2A (0.38) ALDH1A1SMN1; SMN2ALOX5PTGESTRPV1
SCHEMBL8856354 0.78 TRPV1 (0.37) ALDH1A1SMN1; SMN2ALOX5PTGESTRPV1
SCHEMBL8856712 0.78 TLR8 (0.39) ALDH1A1SMN1; SMN2TRPV1L3MBTL1HTT
SCHEMBL8856287 0.78 TRPV1 (0.37) ALDH1A1SMN1; SMN2ALOX5PTGESTRPV1
SCHEMBL8856274 0.77 KMT2A (0.46) ALDH1A1SMN1; SMN2ALOX5TRPV1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5656634-A N-aryl and N-heteroarylamide and urea derivatives as inhibitors of acyl coenzyme A: cholesterol acyl transferase (ACAT) PFIZER INC. (US) 1997-08-12 US disclosed
US-5362878-A Intermediates for making N-aryl and N-heteroarylamide and urea derivatives as inhibitors of acyl coenzyme A: cholesterol acyl transferase (ACAT) PFIZER INC. (US) 1994-11-08 US disclosed