SCHEMBL8859019

SCHEMBL8859019

OCCOCCCN1c2ccccc2CCc2ccccc21

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 10/20 0.61
HTR2A P28223 3/20 0.57
SLC6A2 P23975 3/20 0.53
SLC22A2 O15244 2/20 0.53
SLC22A1 O15245 2/20 0.53
SLC22A3 O75751 2/20 0.53
CHRM2 P08172 2/20 0.53
CYP2D6 P10635 2/20 0.53
CHRM1 P11229 2/20 0.53
DRD2 P14416 2/20 0.53
ADRA2B P18089 2/20 0.53
ADRA2C P18825 2/20 0.53
CHRM3 P20309 2/20 0.53
HTR2C P28335 2/20 0.53
ADRA1A P35348 2/20 0.53
HRH1 P35367 2/20 0.53
DRD3 P35462 2/20 0.53
SCN1A P35498 2/20 0.53
OPRK1 P41145 2/20 0.53
HTR2B P41595 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9083641 0.84 SLC6A1 (0.51) SLC6A4HTR2AMEN1KMT2ASLC6A1
SCHEMBL6961973 0.83 HTR2A (0.68) SLC6A4HTR2ASLC6A2SLC22A2SLC22A1
SCHEMBL7168298 0.82 HTR2A (0.66) SLC6A4HTR2ASLC6A2SLC22A2SLC22A1
SCHEMBL6637686 0.79 HTR2A (0.61) SLC6A4HTR2ASLC6A2SLC22A2SLC22A1
SCHEMBL13051501 0.79 HTR2A (0.78) SLC6A4HTR2ASLC6A2SLC22A2SLC22A1
SCHEMBL14140510 0.79 HTR2A (0.62) SLC6A4HTR2ASLC6A2SLC22A2SLC22A1
SCHEMBL5711008 0.78 ALDH1A1 (0.44) SLC6A4HTR2ASLC6A2CHRM2CHRM1
SCHEMBL8201084 0.77 HTR2A (0.59) SLC6A4HTR2ASLC6A2SLC22A2SLC22A1
SCHEMBL11376146 0.76 HTR2A (0.54) SLC6A4HTR2ASLC6A2SLC22A2SLC22A1
SCHEMBL11376142 0.75 HTR2A (0.57) SLC6A4HTR2ASLC6A2SLC22A2SLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997022342-A1 NOVEL METHOD NOVO NORDISK A/S (DK) 1997-06-26 WO disclosed
EP-0585314-B1 NOVEL HETEROCYCLIC CARBOXYLIC ACIDS NOVO NORDISK AS (DK) 1996-09-18 EP disclosed
US-5348965-A N-substituted azaheterocyclic carboxylic acids NOVO NORDISK A/S (DK) 1994-09-20 US disclosed
EP-0585314-A1 NOVEL HETEROCYCLIC CARBOXYLIC ACIDS. NOVO NORDISK AS (DK) 1994-03-09 EP disclosed
WO-1992020658-A1 NOVEL HETEROCYCLIC CARBOXYLIC ACIDS NOVO NORDISK A/S (DK) 1992-11-26 WO disclosed