SCHEMBL8862099

SCHEMBL8862099

COc1ccc(C#CCCCCCC(C)(C)[Si](O[Si](c2ccccc2)(c2ccccc2)C(C)(C)CCCCCC#Cc2ccc(OC)cc2)(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
MAPT P10636 1/20 0.45
CYP2C9 P11712 1/20 0.45
TSHR P16473 1/20 0.45
CYP2C19 P33261 1/20 0.45
MMP2 P08253 4/20 0.35
MMP3 P08254 3/20 0.35
MMP13 P45452 3/20 0.35
PTPN2 P17706 1/20 0.35
PTPN1 P18031 1/20 0.35
PTPN6 P29350 1/20 0.35
PTPN11 Q06124 1/20 0.35
PPARG P37231 1/20 0.35
PPARD Q03181 1/20 0.35
PPARA Q07869 1/20 0.35
GRIN2B Q13224 1/20 0.34
GBA1 P04062 1/20 0.33
MMP9 P14780 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8862123 1.00 ALDH1A1 (0.45) ALDH1A1CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL8862091 0.79 TDP1 (0.49) ALDH1A1MMP2MMP3MMP1
SCHEMBL8862044 0.79 TDP1 (0.49) ALDH1A1MMP2MMP3MMP1
SCHEMBL8862120 0.76 MAPT (0.47) ALDH1A1CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL8862128 0.76 CYP3A4 (0.33) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8862016 0.76 CYP3A4 (0.33) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL9311733 0.74 CYP3A4 (0.32) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8862098 0.73 MAPT (0.46) ALDH1A1CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL9367547 0.72 CYP3A4 (0.47) ALDH1A1CYP1A2CYP3A4MAPTCYP2C9
SCHEMBL9429436 0.71 FFAR1 (0.49) ALDH1A1CYP1A2CYP3A4MAPTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5656636-A TREATING PSORIASIS SMITHKLINE BEECHAM CORPORATION (US) 1997-08-12 US disclosed
US-5633258-A Pyridine compounds for treating leukotriene-related diseases SMITHKLINE BEECHAM CORPORATION (US) 1997-05-27 US disclosed
US-5631262-A Pyridine compounds for treating leukotriene-related diseases SMITHKLINE BEECHAM CORPORATION (US) 1997-05-20 US disclosed