SCHEMBL886480

SCHEMBL886480

CCCN1C(=O)c2ccccc2C1=O

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GLS O94925 1/20 0.61
DRD3 P35462 1/20 0.58
MEN1 O00255 1/20 0.55
CYP1A2 P05177 1/20 0.55
CHRM2 P08172 1/20 0.55
CYP2C19 P33261 1/20 0.55
KMT2A Q03164 1/20 0.55
NPC1 O15118 1/20 0.53
CASP3 P42574 1/20 0.53
RAB9A P51151 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
SENP8 Q96LD8 1/20 0.53
SENP7 Q9BQF6 1/20 0.53
SENP6 Q9GZR1 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29683253 1.00 GLS (0.61) GLSDRD3MEN1CYP1A2CHRM2
Bromide SCHEMBL17510030 0.98 GLS (0.59) GLSDRD3MEN1CYP1A2CHRM2
SCHEMBL27494119 0.90 GLS (0.52) GLSDRD3CASP3
SCHEMBL29511230 0.87 CHRM2 (0.61) MEN1CYP1A2CHRM2CYP2C19KMT2A
SCHEMBL149620 0.87 CHRM2 (0.61) MEN1CYP1A2CHRM2CYP2C19KMT2A
SCHEMBL5151493 0.86 DRD3 (0.50) GLSDRD3
SCHEMBL10335609 0.86 DRD3 (0.50) GLSDRD3
SCHEMBL6699936 0.85 GLS (0.71) GLSNPC1CASP3RAB9ASMN1; SMN2
SCHEMBL19297268 0.85 ALDH1A1 (0.62) DRD3CHRM2
SCHEMBL29418113 0.85 ALDH1A1 (0.67) MEN1CYP1A2CHRM2CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 382 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114349678-B Continuous industrial production method of N-alkyl-nitrophthalimide 珠海派锐尔新材料有限公司 2024-04-26 CN claimed
CN-114349678-A Continuous industrial production method of N-alkyl-nitrophthalimide 珠海派锐尔新材料有限公司 2022-04-15 CN claimed
CN-110306346-A A kind of refining dye enzyme and preparation method thereof promoting the anti-fuzz balls performance of cotton knitwear 广东湛丰精细化工有限公司 2019-10-08 CN claimed
US-20160311773-A1 GLUCOSE METABOLISM MODULATING COMPOUNDS NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2016-10-27 US claimed
CN-101490334-B Substantially flame retardant-free 3GT carpet DU PONT 2012-09-05 CN claimed
US-20120135089-A1 E3 LIGASE INHIBITORS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2012-05-31 US claimed
US-8148537-B2 Substituted acetophenones useful as PDE4 inhibitors LEO PHARMA A/S (DK) 2012-04-03 US claimed
US-20110118300-A1 GLUCOSE METABOLISM MODULATING COMPOUNDS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-05-19 US claimed
EP-2125736-B1 SUBSTITUTED ACETOPHENONES USEFUL AS PDE4 INHIBITORS LEO PHARMA AS (DK) 2011-03-30 EP claimed
WO-2010107485-A1 E3 LIGASE INHIBITORS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2010-09-23 WO claimed
US-20060069262-A1 Oxadiazoles and their manufacture EASTMAN KODAK COMPANY 2006-03-30 US claimed
US-20030050310-A1 Hydroxamic acid derivatives as proteinase inhibitors BRITISH BIOTECH PHARMACEUTICALS LTD. (GB) 2003-03-13 US claimed
US-6479502-B1 TREATMENT OF DISEASES AND CONDITIONS RESPONSIVE TO MODULATION OF MATRIX METALLOPROTEINASE ACTIVITY BRITISH BIOTECH PHARMACEUTICALS (GB) 2002-11-12 US claimed
EP-1107953-A1 HYDROXAMIC ACID DERIVATIVES AS PROTEINASE INHIBITORS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 2001-06-20 EP claimed
WO-2000012477-A1 HYDROXAMIC ACID DERIVATIVES AS PROTEINASE INHIBITORS BRITISH BIOTECH PHARMACEUTICALS LIMITED (GB) 2000-03-09 WO claimed
US-5719295-A FROM N-ALKYL NITROPHTHALAMIDE GENERAL ELECTRIC COMPANY (US) 1998-02-17 US claimed
US-5688312-A INKS WITH COLORS AND IMIDES OR BISIMIDES, FOR ACOUSTIC INK PRINTER AND DROP EJECTOR XEROX CORPORATION (US) 1997-11-18 US claimed
EP-0164409-B1 METHOD FOR MAKING N-SUBSTITUTED NITROPHTHALIMIDES GENERAL ELECTRIC COMPANY (US) 1989-08-02 EP claimed
EP-0164409-A1 METHOD FOR MAKING N-SUBSTITUTED NITROPHTHALIMIDES. GEN ELECTRIC (US) 1985-12-18 EP claimed
WO-1985002612-A1 METHOD FOR MAKING N-SUBSTITUTED NITROPHTHALIMIDES GENERAL ELECTRIC COMPANY (US) 1985-06-20 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110118300-A1 GLUCOSE METABOLISM MODULATING COMPOUNDS SLC2A4, SLC2A2, SLC2A1 GLS 49/4885DRD3 604/4885MEN1 2600/4885
US-20120135089-A1 E3 LIGASE INHIBITORS MDM2, RBX1, XIAP GLS 2863/4885DRD3 4572/4885MEN1 2333/4885
US-20030050310-A1 Hydroxamic acid derivatives as proteinase inhibitors MMP2, CTSH, TIMP3 GLS 542/4885DRD3 4718/4885MEN1 3457/4885
US-20060069262-A1 Oxadiazoles and their manufacture OXA1L, CYP1B1, OXER1 GLS 2705/4885DRD3 478/4885MEN1 1167/4885
US-20160311773-A1 GLUCOSE METABOLISM MODULATING COMPOUNDS SLC2A4, SLC2A2, SLC2A1 GLS 36/4885DRD3 597/4885MEN1 2768/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.