Formamide

Formamide

SCHEMBL8865992

CC(Cc1cccc(N)c1)c1ccccc1.NC=O

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.46
MAOB P27338 3/20 0.46
NR3C2 P08235 1/20 0.44
ADRB2 P07550 4/20 0.41
TAAR1 Q96RJ0 5/20 0.41
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
CYP2A6 P11509 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
OPRK1 P41145 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CPN1 P15169 1/20 0.38
CPB2 Q96IY4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10351218 0.92 MAOA (0.53) MAOAMAOBNR3C2ADRB2TAAR1
Formamide SCHEMBL7267893 0.85 TAAR1 (0.50) MAOANR3C2TAAR1SLC6A2SLC6A4
SCHEMBL310745 0.85 ADRB2 (0.48) MAOAMAOBADRB2TAAR1SLC6A2
SCHEMBL30495002 0.85 ADRB2 (0.48) MAOAMAOBADRB2TAAR1SLC6A2
SCHEMBL3260417 0.84 ADRB2 (0.50) MAOAMAOBADRB2TAAR1SLC6A2
SCHEMBL7930021 0.84 ADRB2 (0.47) MAOAMAOBADRB2TAAR1SLC6A2
Formamide SCHEMBL8865892 0.84 PNMT (0.57) MAOANR3C2TAAR1SLC6A2SLC6A4
SCHEMBL28087034 0.82 CYP19A1 (0.52) MAOAMAOBADRB2TAAR1SLC6A2
SCHEMBL8580067 0.82 MAOA (0.52) MAOAMAOBADRB2TAAR1SLC6A2
SCHEMBL1099930 0.80 ADRB2 (0.47) MAOAMAOBADRB2TAAR1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5605916-A Arylalkyl-amines having anticonvulsant and neuroprotective properties ASTRA AB (SE) 1997-02-25 US disclosed
US-5539120-A Arylalkyl-amines having anticonvulsant and neuroprotective properties AGENCE SPATIALE EUROPEENNE (FR) 1996-07-23 US disclosed
EP-0356035-B1 Arylkalkyl-amines and -amides having anticonvulsant and neuroprotective properties ASTRA AB (SE) 1996-03-13 EP disclosed
US-5430044-A Arylalkyl-amines and -amides having anticonvulsant and neuroprotective properties FISONS CORPORATION (GB) 1995-07-04 US disclosed
EP-0648745-A1 Arylalkylamine having anticonvulsant and neuroprotective properties Astra Aktiebolag (SE) 1995-04-19 EP disclosed
EP-0648489-A1 Arylalkylamides having neuroprotective properties FISONS CORPORATION (US) 1995-04-19 EP disclosed
US-5331007-A Arylalkyl-amines and -amides having anticonvulsant and neuroprotective properties FISONS CORPORATION (US) 1994-07-19 US disclosed
WO-1991011995-A1 ARYLALKYL-AMINES AND -AMIDES HAVING ANTICONVULSANT AND NEUROPROTECTIVE PROPERTIES FISONS CORPORATION (US) 1991-08-22 WO disclosed
EP-0356035-A2 Arylkalkyl-amines and -amides having anticonvulsant and neuroprotective properties Astra Aktiebolag (SE) 1990-02-28 EP disclosed