SCHEMBL8866491

SCHEMBL8866491

Clc1cccc2c1C(c1c[nH]cn1)CCC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.38
HTR2C P28335 2/20 0.37
OPRM1 P35372 2/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
OPRL1 P41146 1/20 0.35
ADRA2A P08913 3/20 0.35
ADRA1A P35348 2/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1B P35368 1/20 0.35
KCNN1 Q92952 1/20 0.33
KCNN2 Q9H2S1 1/20 0.33
KCNN3 Q9UGI6 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
CXCR4 P61073 1/20 0.33
HTR2B P41595 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.32
TAS1R1 Q7RTX1 1/20 0.32
TAS1R2 Q8TE23 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8865654 0.84 SLC6A2 (0.35) OPRM1ADRA2AADRA1AADRA1DADRA1B
SCHEMBL8865718 0.81 SRD5A1 (0.39) HTR2COPRM1ADRA2AADRA1AADRA1D
SCHEMBL7608212 0.81 ADRA2A (0.40) HTR2COPRM1OPRD1OPRK1OPRL1
SCHEMBL8865945 0.81 HTR1A (0.41) HTR1A
SCHEMBL769063 0.79 ADRA1A (0.55) OPRM1ADRA2AADRA1AADRA1DADRA1B
SCHEMBL8865200 0.78 ESR1 (0.44) ADRA2AADRA1AADRA1DADRA1B
SCHEMBL8866107 0.78 HTR1A (0.34) HTR2COPRM1ADRA2AADRA1AADRA1D
SCHEMBL7607563 0.76 HTR1A (0.39) HTR2CHTR2BHTR1A
SCHEMBL8865117 0.76 SRD5A1 (0.39) OPRM1ADRA2AADRA1AADRA1DADRA1B
SCHEMBL30543392 0.75 ADRA2A (0.58) P2RX7ADRA2AADRA1AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658938-A HYPOTENSIVE AGENT, ANTIISCHMIC AGENTS U C B S.A. (BE) 1997-08-19 US disclosed
EP-0717037-A1 Substituted 1H-imidazoles having alpha 2-agonistic and alpha 1-antagonistic activity U C B, S.A. (BE) 1996-06-19 EP disclosed