SCHEMBL8865718

SCHEMBL8865718

Clc1ccc2c(c1)CCCC2c1c[nH]cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 4/20 0.39
SRD5A2 P31213 2/20 0.38
ADRA2A P08913 2/20 0.37
ADRA1A P35348 2/20 0.37
ADRA1D P25100 1/20 0.37
ADRA1B P35368 1/20 0.37
HTR2C P28335 2/20 0.37
HTR2A P28223 1/20 0.37
HTR2B P41595 1/20 0.37
FNTA P49354 1/20 0.36
FNTB P49356 1/20 0.36
CYP17A1 P05093 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP11B2 P19099 1/20 0.36
PFKFB3 Q16875 1/20 0.35
FADS1 O60427 1/20 0.35
HTR1A P08908 1/20 0.35
OPRM1 P35372 1/20 0.35
CYP2D6 P10635 1/20 0.35
PYGL P06737 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8865200 0.86 ESR1 (0.44) ADRA2AADRA1AADRA1DADRA1BCYP17A1
SCHEMBL8865117 0.84 SRD5A1 (0.39) SRD5A1ADRA2AADRA1AADRA1DADRA1B
SCHEMBL769063 0.81 ADRA1A (0.55) ADRA2AADRA1AADRA1DADRA1BHTR1A
SCHEMBL8866491 0.81 P2RX7 (0.38) ADRA2AADRA1AADRA1DADRA1BHTR2C
SCHEMBL8865285 0.81 GID4 (0.50) SRD5A1HTR2C
SCHEMBL7614024 0.79 ESR2 (0.42)
Hydrochloric Acid SCHEMBL8865538 0.78 ESR2 (0.41)
SCHEMBL8865311 0.78 ALOX15 (0.51) ADRA2AADRA1AADRA1DADRA1BCYP17A1
SCHEMBL8865423 0.78 KDM4C (0.41) KDM4C
Hydrochloric Acid SCHEMBL8865276 0.77 ALOX15 (0.50) ADRA2AADRA1AADRA1DADRA1BCYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658938-A HYPOTENSIVE AGENT, ANTIISCHMIC AGENTS U C B S.A. (BE) 1997-08-19 US disclosed
EP-0717037-A1 Substituted 1H-imidazoles having alpha 2-agonistic and alpha 1-antagonistic activity U C B, S.A. (BE) 1996-06-19 EP disclosed