SCHEMBL8869461

SCHEMBL8869461

CC(NC(=O)OC(C)(C)C)c1c[nH]c2ccc(Oc3cccnc3)cc12

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.44
CYP3A4 P08684 5/20 0.41
NR4A2 P43354 1/20 0.41
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
THRA P10827 5/20 0.39
THRB P10828 5/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
KIF20A O95235 1/20 0.38
DYRK1A Q13627 1/20 0.38
LMNA P02545 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8869778 0.85 SCN9A (0.45) SCN9ANR4A2MTNR1AMTNR1BTHRA
SCHEMBL8868878 0.85 MTNR1A (0.50) SCN9ANR4A2MTNR1AMTNR1BTHRA
SCHEMBL6226884 0.80 LMNA (0.47) CYP3A4DYRK1ALMNATDP1
SCHEMBL6226878 0.80 LMNA (0.47) CYP3A4DYRK1ALMNATDP1
SCHEMBL8869454 0.79 LTA4H (0.57) CYP3A4MTNR1AMTNR1BTDP1
SCHEMBL8870222 0.79 MTNR1A (0.43) SCN9ACYP3A4NR4A2MTNR1AMTNR1B
SCHEMBL9210783 0.78 LMNA (0.48) MTNR1AMTNR1BKIF20ADYRK1ALMNA
SCHEMBL28007326 0.77 MAP2K1 (0.47) CYP3A4MTNR1ATP53MAPT
SCHEMBL9204210 0.76 LMNA (0.46) NR4A2MTNR1AMTNR1BTHRATHRB
SCHEMBL8883939 0.73 TACR1 (0.41) MTNR1AMTNR1BTHRATHRBTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5637593-A MIGRAINE; HYPOTENSIVE AGENTS SMITHKLINE BEECHAM PLC (GB) 1997-06-10 US disclosed