SCHEMBL8869895

SCHEMBL8869895

COc1ccnc(Oc2ccc3[nH]cc(CC(OC(=O)C(=O)OC(Cc4c[nH]c5ccc(Oc6nccc(OC)n6)cc45)N(C)C)N(C)C)c3c2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 5/20 0.44
CYP1A2 P05177 5/20 0.44
CYP3A4 P08684 4/20 0.44
USP2 O75604 3/20 0.44
CYP2C19 P33261 3/20 0.44
CLK4 Q9HAZ1 3/20 0.44
LMNA P02545 2/20 0.44
KMT2A Q03164 3/20 0.44
HTR2B P41595 4/20 0.43
HTR1A P08908 3/20 0.43
HTR2A P28223 2/20 0.43
HTR2C P28335 2/20 0.43
KDM4E B2RXH2 2/20 0.43
MTNR1A P48039 4/20 0.41
MTNR1B P49286 4/20 0.41
HTR1D P28221 2/20 0.41
HTR1B P28222 2/20 0.41
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8869627 0.83 HTR2B (0.51) CYP2D6CYP1A2CYP3A4KMT2AHTR2B
SCHEMBL8869901 0.81 CYP1A2 (0.51) CYP2D6CYP1A2CYP3A4USP2CYP2C19
Oxalic Acid SCHEMBL8869885 0.81 KMT2A (0.71) CYP2D6CYP1A2CYP3A4USP2CYP2C19
SCHEMBL8868790 0.80 HTR1D (0.67) CYP2D6CYP1A2KMT2AHTR2BHTR1A
SCHEMBL8870342 0.80 SCN9A (0.46) KMT2AHTR2BHTR1AHTR2AHTR2C
SCHEMBL8868849 0.79 SCN9A (0.43) CYP2D6CYP1A2CYP3A4USP2CYP2C19
SCHEMBL8870092 0.79 HTR1D (0.44) KMT2AHTR2BHTR1AHTR2AHTR2C
SCHEMBL8868838 0.77 GPR84 (0.47) CYP2D6CYP1A2CYP3A4USP2CYP2C19
SCHEMBL9204127 0.77 HTR2B (0.45) CYP2D6CYP1A2CYP3A4USP2CYP2C19
SCHEMBL23927939 0.76 HTR2B (0.55) CYP2D6CYP1A2CYP3A4KMT2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5637593-A MIGRAINE; HYPOTENSIVE AGENTS SMITHKLINE BEECHAM PLC (GB) 1997-06-10 US disclosed