SCHEMBL8870092

SCHEMBL8870092

CN(C)C(Cc1c[nH]c2ccc(Oc3ccc(Br)cc3)cc12)OC(=O)C(=O)OC(Cc1c[nH]c2ccc(Oc3ccc(Br)cc3)cc12)N(C)C

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 4/20 0.44
HTR1B P28222 3/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
SCN9A Q15858 4/20 0.44
HTR1A P08908 2/20 0.43
HTR2A P28223 2/20 0.42
HTR2C P28335 1/20 0.42
HTR2B P41595 1/20 0.42
KDM4E B2RXH2 1/20 0.42
TRPM8 Q7Z2W7 1/20 0.41
ADAM17 P78536 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8870342 0.90 SCN9A (0.46) HTR1DHTR1BKMT2ASCN9AHTR1A
SCHEMBL8869627 0.90 HTR2B (0.51) HTR1DHTR1BKMT2AMEN1HTR1A
SCHEMBL8868849 0.84 SCN9A (0.43) HTR1DHTR1BKMT2AMEN1SCN9A
SCHEMBL8868679 0.82 TRPV1 (0.42) HTR1DHTR1BKMT2ASCN9AHTR1A
SCHEMBL8869895 0.79 CYP2D6 (0.44) HTR1DHTR1BKMT2AMEN1HTR1A
SCHEMBL23927939 0.76 HTR2B (0.55) HTR1DHTR1BKMT2AMEN1HTR1A
Oxalic Acid SCHEMBL8870089 0.76 KMT2A (0.73) HTR1DHTR1BKMT2AHTR1AHTR2A
SCHEMBL8868429 0.75 GABRA1 (0.48) KMT2AMEN1KDM4E
SCHEMBL8869175 0.75 HTR1D (0.70) HTR1DHTR1BKMT2AHTR1AHTR2A
SCHEMBL9208221 0.71 HTR2A (0.44) HTR1DHTR1BHTR1AHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5637593-A MIGRAINE; HYPOTENSIVE AGENTS SMITHKLINE BEECHAM PLC (GB) 1997-06-10 US disclosed