SCHEMBL8869901

SCHEMBL8869901

COc1ccnc(Oc2ccc3[nH]cc(CN(C)C)c3c2)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 7/20 0.51
CYP2D6 P10635 7/20 0.51
HTR6 P50406 3/20 0.51
HTR1A P08908 3/20 0.51
HTR2B P41595 2/20 0.51
HTR1D P28221 2/20 0.51
HTR1B P28222 2/20 0.51
HTR2A P28223 2/20 0.51
HTR2C P28335 2/20 0.51
HTR7 P34969 2/20 0.51
HTR4 Q13639 2/20 0.51
MTNR1A P48039 2/20 0.51
HTR3E A5X5Y0 1/20 0.51
HTR3B O95264 1/20 0.51
CYP2C9 P11712 1/20 0.51
HTR1E P28566 1/20 0.51
HTR1F P30939 1/20 0.51
HTR3A P46098 1/20 0.51
HTR5A P47898 1/20 0.51
MTNR1B P49286 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8868790 0.89 HTR1D (0.67) CYP1A2CYP2D6HTR6HTR1AHTR2B
SCHEMBL8869498 0.85 CYP2D6 (0.52) CYP1A2CYP2D6HTR6HTR1AHTR2B
Oxalic Acid SCHEMBL8869885 0.84 KMT2A (0.71) CYP1A2CYP2D6HTR6HTR1AHTR2B
SCHEMBL8868838 0.84 GPR84 (0.47) CYP1A2CYP2D6HTR6HTR1AHTR2B
SCHEMBL8869895 0.81 CYP2D6 (0.44) CYP1A2CYP2D6HTR6HTR1AHTR2B
SCHEMBL1196012 0.81 HTR2A (0.74) CYP1A2CYP2D6HTR6HTR1AHTR2B
SCHEMBL9204127 0.80 HTR2B (0.45) CYP1A2CYP2D6HTR6HTR1AHTR2B
SCHEMBL8869870 0.79 HTR1A (0.63) CYP1A2CYP2D6HTR6HTR1AHTR2B
SCHEMBL8870217 0.76 MTNR1A (0.55) CYP1A2CYP2D6HTR1AHTR2BMTNR1A
SCHEMBL11258933 0.74 HTR1D (0.56) CYP1A2CYP2D6HTR6HTR1AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5637593-A MIGRAINE; HYPOTENSIVE AGENTS SMITHKLINE BEECHAM PLC (GB) 1997-06-10 US disclosed