SCHEMBL8870342

SCHEMBL8870342

Cc1ccc(Oc2ccc3[nH]cc(CC(OC(=O)C(=O)OC(Cc4c[nH]c5ccc(Oc6ccc(C)cc6)cc45)N(C)C)N(C)C)c3c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 3/20 0.46
HTR1D P28221 4/20 0.45
HTR1B P28222 3/20 0.45
HTR1A P08908 2/20 0.43
KMT2A Q03164 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43
KDM4E B2RXH2 1/20 0.43
P2RY14 Q15391 1/20 0.42
TRPM8 Q7Z2W7 1/20 0.42
TACR1 P25103 1/20 0.41
LTA4H P09960 1/20 0.41
PLA2G2A P14555 1/20 0.41
ICMT O60725 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8869627 0.91 HTR2B (0.51) HTR1DHTR1BHTR1AKMT2AHTR2A
SCHEMBL8870092 0.90 HTR1D (0.44) SCN9AHTR1DHTR1BHTR1AKMT2A
SCHEMBL8868849 0.85 SCN9A (0.43) SCN9AHTR1DHTR1BHTR1AKMT2A
SCHEMBL8868679 0.83 TRPV1 (0.42) SCN9AHTR1DHTR1BHTR1AKMT2A
SCHEMBL8869895 0.80 CYP2D6 (0.44) HTR1DHTR1BHTR1AKMT2AHTR2A
SCHEMBL23927939 0.77 HTR2B (0.55) HTR1DHTR1BHTR1AKMT2AHTR2A
SCHEMBL8870437 0.76 HTR1D (0.52) HTR1DHTR1BHTR1AKMT2AHTR2A
SCHEMBL8868429 0.76 GABRA1 (0.48) KMT2AKDM4ETACR1LTA4HPLA2G2A
Oxalic Acid SCHEMBL8870335 0.76 KMT2A (0.75) HTR1DHTR1BHTR1AKMT2AHTR2A
SCHEMBL8869593 0.74 HTR1D (0.71) HTR1DHTR1BHTR1AKMT2AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5637593-A MIGRAINE; HYPOTENSIVE AGENTS SMITHKLINE BEECHAM PLC (GB) 1997-06-10 US disclosed