SCHEMBL8870033

SCHEMBL8870033

O=c1sc2ccc(Cl)cc2n1CCCCl

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 3/20 0.67
SIGMAR1 Q99720 1/20 0.59
HTR1A P08908 2/20 0.47
HTR7 P34969 2/20 0.47
RAB9A P51151 3/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
NPC1 O15118 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MAPT P10636 1/20 0.45
ALPG P10696 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
CNR2 P34972 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15295194 0.87 TMEM97 (0.66) TMEM97SIGMAR1HTR1AHTR7CNR2
SCHEMBL8870438 0.87 TMEM97 (0.66) TMEM97SIGMAR1HTR1AHTR7RAB9A
SCHEMBL15283315 0.84 TMEM97 (0.63) TMEM97SIGMAR1HTR1AHTR7RAB9A
SCHEMBL9570355 0.83 TMEM97 (0.62) TMEM97SIGMAR1HTR1AHTR7RAB9A
SCHEMBL15292530 0.83 TMEM97 (0.62) TMEM97SIGMAR1HTR1AHTR7RAB9A
SCHEMBL9570335 0.83 SIGMAR1 (0.71) TMEM97SIGMAR1HTR1AHTR7RAB9A
Iodide SCHEMBL8869500 0.82 TMEM97 (0.60) TMEM97SIGMAR1HTR1AHTR7RAB9A
Hydrochloric Acid SCHEMBL8869860 0.82 SIGMAR1 (0.69) TMEM97SIGMAR1HTR1AHTR7CYP1A2
SCHEMBL318427 0.80 L3MBTL1 (0.68) SIGMAR1RAB9AL3MBTL1NPC1CYP1A2
SCHEMBL3225943 0.79 HTT (0.65) TMEM97SIGMAR1L3MBTL1CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5654323-A 2-NITROGEN-CONTAINING FUNCTIONAL GROUP-HALOBENZOTHIAZOLES; ANALGESICS; ANTIINFLAMMATORY AND HYPOTENSIVE AGENTS; INHIBITORS OF CYTOKINES (INCLUDING TUMOR NECROSIS FACTOR) AND PHOSPHOLIPASE; SEPTIC SHOCK ADIR ET COMPAGNIE (FR) 1997-08-05 US disclosed
US-5597819-A ANTIINFLAMMATORY AGENTS ADIR ET COMPAGNIE (FR) 1997-01-28 US disclosed
US-5550143-A Heterocyclic compounds ADIR ET COMPAGNIE (FR) 1996-08-27 US disclosed
EP-0572308-A2 Heterocyclic derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1993-12-01 EP disclosed