SCHEMBL8871022

SCHEMBL8871022

N#Cc1ccc2[nH]c(C3=CCN(CCCCc4c[nH]c5ccc(C#N)cc45)CC3)cc2c1

nearest known ligand 0.59

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 6/20 0.58
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
MAPT P10636 1/20 0.56
CYP2C9 P11712 1/20 0.56
DRD2 P14416 1/20 0.56
TSHR P16473 1/20 0.56
DRD4 P21917 1/20 0.56
CYP2C19 P33261 1/20 0.56
DRD3 P35462 1/20 0.56
TDP1 Q9NUW8 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8871408 0.90 TDP1 (0.58) HTR1ACYP1A2CYP3A4MAPTCYP2C9
SCHEMBL9229535 0.88 SLC6A4 (0.64) HTR1ACYP1A2CYP3A4MAPTCYP2C9
SCHEMBL9581909 0.87 HTR1A (0.74) HTR1ACYP1A2CYP3A4MAPTCYP2C9
SCHEMBL8870806 0.84 HTR1A (0.59) HTR1ACYP1A2CYP3A4MAPTCYP2C9
SCHEMBL11115378 0.83 HTR1A (0.56) HTR1ACYP1A2CYP3A4MAPTCYP2C9
SCHEMBL8871095 0.82 HTR1A (0.61) HTR1ACYP1A2CYP3A4MAPTCYP2C9
SCHEMBL8871306 0.81 HTR1A (0.77) HTR1ACYP1A2CYP3A4MAPTCYP2C9
SCHEMBL8552552 0.80 KDM4E (0.62) HTR1ADRD2DRD4DRD3TDP1
SCHEMBL8555864 0.80 KDM4E (0.62) HTR1ADRD2DRD4DRD3TDP1
SCHEMBL8871147 0.79 HTR1A (0.59) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5693655-A 3-indolylpiperidines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-02 US disclosed