SCHEMBL8872298

SCHEMBL8872298

COC(=O)c1ccccc1-c1ccc(COS(=O)(=O)c2ccc(C)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 4/20 0.50
SLC6A4 P31645 3/20 0.50
SLC6A2 P23975 1/20 0.45
BCL2L1 Q07817 1/20 0.44
FFAR4 Q5NUL3 1/20 0.44
LTB4R2 Q9NPC1 1/20 0.43
BDKRB1 P46663 4/20 0.43
KMT2A Q03164 3/20 0.42
BRS3 P32247 1/20 0.42
MAPT P10636 1/20 0.41
MEN1 O00255 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8871657 0.92 SLC6A3 (0.53) SLC6A3SLC6A4SLC6A2BCL2L1LTB4R2
SCHEMBL8873455 0.90 LMNA (0.50) BCL2L1LTB4R2KMT2AMAPTMEN1
SCHEMBL8873666 0.83 SLC6A3 (0.57) SLC6A3SLC6A4SLC6A2BCL2L1LTB4R2
SCHEMBL8872457 0.82 TSHR (0.48) BCL2L1LTB4R2KMT2AMAPTMEN1
SCHEMBL8874327 0.82 SLC6A3 (0.56) SLC6A3SLC6A4SLC6A2BCL2L1LTB4R2
SCHEMBL8873311 0.82 KMT2A (0.58) KMT2AMAPT
SCHEMBL8971371 0.81 SLC6A3 (0.52) SLC6A3SLC6A4SLC6A2BCL2L1LTB4R2
SCHEMBL249 0.81 SLC6A3 (0.73) SLC6A3SLC6A4SLC6A2LTB4R2MAPT
SCHEMBL5870583 0.80 KMT2A (0.62) KMT2AMAPT
SCHEMBL8872453 0.78 CA12 (0.59) BCL2L1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587504-A Sulfonyloxy-biphenylcarboxylic ester derivatives which are intermediates EISAI CO., LTD. (JP) 1996-12-24 US claimed
US-5700938-A Intermediates for imidazopyridine derivatives EISAI CO., LTD. (JP) 1997-12-23 US disclosed
US-5618969-A Intermediates for imidazopyridines EISAI CO., LTD. (JP) 1997-04-08 US disclosed
US-5608068-A Process for the preparation of imidazopyridine derivatives and intermediates EISAI CO., LTD. (JP) 1997-03-04 US disclosed
US-5587504-A Sulfonyloxy-biphenylcarboxylic ester derivatives which are intermediates EISAI CO., LTD. (JP) 1996-12-24 US disclosed
US-5583229-A Process for the preparation of imidazopyridine derivatives EISAI CO., LTD. (JP) 1996-12-10 US disclosed
US-5559236-A Intermediates for substituted biphenylmethylmidazopyridine angiotensin II antagonists EISAI CO., LTD. (JP) 1996-09-24 US disclosed
US-5557002-A Process for the preparation of biphenyl containing intermediates useful in making angiotensin II receptor antagonists EISAI CO., LTD. (JP) 1996-09-17 US disclosed
US-5554757-A Process for the preparation of imidazopyridine derivatives, and intermediates therefore EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0627433-A1 PROCESS FOR PRODUCING IMIDAZOPYRIDINE DERIVATIVE AND INTERMEDIATE Eisai Co., Ltd. (JP) 1994-12-07 EP disclosed