SCHEMBL8875415

SCHEMBL8875415

Cc1ccccc1N1CCN(CC(=O)c2cccc3c(=O)c(C)c(-c4ccccc4)oc23)CC1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.61
LMNA P02545 5/20 0.60
ALDH1A1 P00352 4/20 0.60
NPSR1 Q6W5P4 3/20 0.60
MAPT P10636 3/20 0.60
HTR1A P08908 6/20 0.58
ADRA1A P35348 6/20 0.58
ADRA1D P25100 5/20 0.58
ADRA1B P35368 5/20 0.58
KDM4E B2RXH2 1/20 0.54
CYP1A2 P05177 1/20 0.54
CHRM2 P08172 1/20 0.54
CYP3A4 P08684 1/20 0.54
ADRA2A P08913 1/20 0.54
ADORA3 P0DMS8 1/20 0.54
CYP2D6 P10635 1/20 0.54
CHRM1 P11229 1/20 0.54
ACHE P22303 1/20 0.54
SLC6A2 P23975 1/20 0.54
PDE4A P27815 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8875705 0.99 SMN1; SMN2 (0.61) SMN1; SMN2LMNAALDH1A1NPSR1MAPT
SCHEMBL8874797 0.89 ALDH1A1 (0.76) SMN1; SMN2LMNAALDH1A1NPSR1MAPT
Hydrochloric Acid SCHEMBL8876184 0.88 ALDH1A1 (0.75) SMN1; SMN2LMNAALDH1A1NPSR1MAPT
SCHEMBL8876945 0.88 LMNA (0.64) SMN1; SMN2LMNAALDH1A1NPSR1MAPT
Hydrochloric Acid SCHEMBL8876370 0.87 LMNA (0.63) SMN1; SMN2LMNAALDH1A1NPSR1MAPT
SCHEMBL8876371 0.81 HTR1A (0.76) SMN1; SMN2LMNAALDH1A1NPSR1MAPT
SCHEMBL8877620 0.80 SMN1; SMN2 (0.51) SMN1; SMN2LMNAALDH1A1NPSR1MAPT
Hydrochloric Acid SCHEMBL8875494 0.80 HTR1A (0.75) SMN1; SMN2LMNAALDH1A1NPSR1MAPT
Hydrochloric Acid SCHEMBL8876083 0.80 SMN1; SMN2 (0.51) SMN1; SMN2LMNAALDH1A1NPSR1MAPT
SCHEMBL8876229 0.79 HTR1A (0.79) SMN1; SMN2LMNAALDH1A1HTR1AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5605896-A Bicyclic heterocyclic derivatives having α1 adrenergic and 5HT1A activities RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1997-02-25 US claimed
US-5403842-A Adrenergic blocking and antiserotonine agents; urogenital disorders including spasms of the urethral tract and prostrate problems RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1995-04-04 US claimed
EP-0558245-A1 Heterobicyclic compounds as antagogists of alpha-1 adrenergic and SHT1A receptors RECORDATI S.A. CHEMICAL and PHARMACEUTICAL COMPANY (CH) 1993-09-01 EP claimed