SCHEMBL8877620

SCHEMBL8877620

Cc1ccccc1N1CCN(CC(O)c2cccc3c(=O)c(C)c(-c4ccccc4)oc23)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.51
LMNA P02545 3/20 0.51
ALDH1A1 P00352 3/20 0.51
NPSR1 Q6W5P4 2/20 0.51
MAPT P10636 1/20 0.51
ADRA1A P35348 7/20 0.49
ADRA1D P25100 6/20 0.49
ADRA1B P35368 6/20 0.49
HTR1A P08908 4/20 0.49
KDM4E B2RXH2 1/20 0.47
CYP1A2 P05177 1/20 0.47
CHRM2 P08172 1/20 0.47
CYP3A4 P08684 1/20 0.47
ADRA2A P08913 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
CYP2D6 P10635 1/20 0.47
CHRM1 P11229 1/20 0.47
ACHE P22303 1/20 0.47
SLC6A2 P23975 1/20 0.47
PDE4A P27815 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8876083 0.99 SMN1; SMN2 (0.51) SMN1; SMN2LMNAALDH1A1NPSR1MAPT
SCHEMBL8875644 0.89 LMNA (0.65) SMN1; SMN2LMNAALDH1A1MAPTADRA1A
SCHEMBL8875106 0.89 ALDH1A1 (0.55) SMN1; SMN2LMNAALDH1A1ADRA1AADRA1D
Hydrochloric Acid SCHEMBL8876509 0.89 LMNA (0.64) SMN1; SMN2LMNAALDH1A1MAPTADRA1A
Hydrochloric Acid SCHEMBL8875096 0.88 ALDH1A1 (0.54) SMN1; SMN2LMNAALDH1A1ADRA1AADRA1D
SCHEMBL8877659 0.81 HTR1A (0.65) LMNAALDH1A1ADRA1AADRA1DADRA1B
SCHEMBL8875415 0.80 SMN1; SMN2 (0.61) SMN1; SMN2LMNAALDH1A1NPSR1MAPT
Hydrochloric Acid SCHEMBL8877171 0.80 HTR1A (0.65) LMNAALDH1A1ADRA1AADRA1DADRA1B
SCHEMBL8875442 0.80 HTR1A (0.69) LMNAALDH1A1ADRA1AADRA1DADRA1B
Hydrochloric Acid SCHEMBL8875705 0.80 SMN1; SMN2 (0.61) SMN1; SMN2LMNAALDH1A1NPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1040434-C Heterobicyclic compounds RECORDATI CHEM PHARM (CH) 1998-10-28 CN claimed
US-5605896-A Bicyclic heterocyclic derivatives having α1 adrenergic and 5HT1A activities RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1997-02-25 US claimed
US-5403842-A Adrenergic blocking and antiserotonine agents; urogenital disorders including spasms of the urethral tract and prostrate problems RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1995-04-04 US claimed
WO-1993017007-A1 HETEROBICYCLIC COMPOUNDS RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA S.P.A. (IT) 1993-09-02 WO claimed
EP-0558245-A1 Heterobicyclic compounds as antagogists of alpha-1 adrenergic and SHT1A receptors RECORDATI S.A. CHEMICAL and PHARMACEUTICAL COMPANY (CH) 1993-09-01 EP claimed