SCHEMBL8875425

SCHEMBL8875425

COc1ccccc1N1CCN(CC(C)(C)CO)CC1

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.59
DRD3 P35462 4/20 0.57
ADRA1D P25100 2/20 0.56
ADRA1A P35348 2/20 0.56
ADRA1B P35368 2/20 0.56
HTR1A P08908 1/20 0.56
KDM4E B2RXH2 3/20 0.54
MAPK1 P28482 2/20 0.54
LMNA P02545 1/20 0.54
HTT P42858 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
HTR7 P34969 2/20 0.54
DRD4 P21917 2/20 0.54
HRH1 P35367 2/20 0.54
ALDH1A1 P00352 1/20 0.53
KMT2A Q03164 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
HRH2 P25021 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8980652 0.99 DRD2 (0.58) DRD2DRD3ADRA1DADRA1AADRA1B
SCHEMBL8877466 0.86 DRD2 (0.59) DRD2DRD3ADRA1DADRA1AADRA1B
SCHEMBL8877327 0.86 DRD2 (0.62) DRD2DRD3ADRA1DADRA1AADRA1B
SCHEMBL13254564 0.85 DRD2 (0.66) DRD2DRD3ADRA1DADRA1AADRA1B
SCHEMBL7830825 0.83 ADRA1A (0.62) DRD2DRD3ADRA1DADRA1AADRA1B
SCHEMBL1387894 0.83 DRD2 (0.62) DRD2DRD3ADRA1DADRA1AADRA1B
SCHEMBL1193073 0.80 DRD2 (0.75) DRD2DRD3ADRA1DADRA1AADRA1B
SCHEMBL9126731 0.80 DRD2 (0.58) DRD2DRD3ADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL8875492 0.78 DRD2 (0.57) DRD2DRD3ADRA1DADRA1AADRA1B
SCHEMBL8521957 0.78 HTR1A (0.57) DRD2DRD3HTR1AKDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5605896-A Bicyclic heterocyclic derivatives having α1 adrenergic and 5HT1A activities RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1997-02-25 US disclosed
US-5474994-A Treating hypertension, urethral and lower urinary tract contractions RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1995-12-12 US disclosed