SCHEMBL8877441

SCHEMBL8877441

CCOC(=O)Cc1c(C)n(Cc2ccc(Br)cc2)c2ccc(OC)cc12

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.79
LMNA P02545 2/20 0.64
CYP1A2 P05177 2/20 0.64
CYP3A4 P08684 2/20 0.64
CYP2C9 P11712 2/20 0.64
TSHR P16473 2/20 0.64
CYP2C19 P33261 2/20 0.64
PMP22 Q01453 2/20 0.64
MEN1 O00255 1/20 0.64
RGS12 O14924 1/20 0.64
ALDH1A1 P00352 1/20 0.64
MAPT P10636 1/20 0.64
PKM P14618 1/20 0.64
NFKB1 P19838 1/20 0.64
MAPK1 P28482 1/20 0.64
GNAI1 P63096 1/20 0.64
KMT2A Q03164 1/20 0.64
HIF1A Q16665 1/20 0.64
PLA2G2A P14555 5/20 0.64
PLA2G1B P04054 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8296317 0.94 LMNA (0.69) PTGS2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL8607520 0.92 PTGS2 (0.82) PTGS2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL8292280 0.91 LMNA (0.78) PTGS2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL8296825 0.91 LMNA (0.66) PTGS2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL8949489 0.90 PTGS2 (0.63) PTGS2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL7962081 0.89 PLA2G2A (0.80) PTGS2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL8875901 0.89 PTGS2 (0.68) PTGS2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL8607505 0.88 PTGS2 (1.00) PTGS2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL8292089 0.88 PLA2G2A (0.64) PTGS2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL8610794 0.87 PTGS2 (0.82) PTGS2LMNACYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5639780-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS MERCK FROSST CANADA, INC. (CA) 1997-06-17 US disclosed
WO-1996037467-A1 N-BENZYLINDOL-3-YL BUTANOIC ACID DERIVATIVES AS CYCLOOXYGENASE-2 INHIBITORS MERCK FROSST CANADA INC. (CA) 1996-11-28 WO disclosed