SCHEMBL8879834

SCHEMBL8879834

CCC(O)c1cc(Br)no1

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 6/20 0.44
ADRB1 P08588 6/20 0.44
ADRB3 P13945 5/20 0.44
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10341872 0.85 ADRB2 (0.45) ADRB2ADRB1ADRB3
SCHEMBL6074550 0.84 ADRB2 (0.39) ADRB2ADRB1ADRB3LMNA
SCHEMBL8129014 0.83 ADRB2 (0.40) ADRB2ADRB1ADRB3
SCHEMBL6074317 0.83 ADRB2 (0.40) ADRB2ADRB1ADRB3
SCHEMBL5789095 0.78 ALDH1A1 (0.40) LMNA
SCHEMBL21009819 0.78 ALDH1A1 (0.40) LMNA
SCHEMBL4538650 0.77 ADRB2 (0.54) ADRB2ADRB1ADRB3LMNA
SCHEMBL3439382 0.76 ADRB2 (0.33) ADRB2ADRB1ADRB3
SCHEMBL3466377 0.76 ADRB2 (0.33) ADRB2ADRB1ADRB3
SCHEMBL5791247 0.76 LMNA (0.33) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5602160-A MUSCLE RELAXANT MITSUI TOATSU CHEMICALS INCORPORATED (JP) 1997-02-11 US disclosed
US-5498619-A MUSCLE RELAXANTS, POLLAKIUREA CURING AGENTS AND MUSCLE SPASMS MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1996-03-12 US disclosed
EP-0414391-B1 Aminoketone derivatives and use thereof MITSUI TOATSU CHEMICALS (JP) 1995-03-15 EP disclosed
US-5338857-A Muscle relaxant MITSUI TOATSU CHEMICALS INCORPORATED (JP) 1994-08-16 US disclosed
EP-0414391-A2 Aminoketone derivatives and use thereof MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-02-27 EP disclosed
EP-0207955-B1 PROCESS FOR THE PREPARATION OF 3,5-DISUBSTITUTED ISOXAZOLES ZAMBON S.p.A. (IT) 1990-02-07 EP disclosed
US-4772719-A FROM DIHALOFORMALDOXIME AND ALKYNE, CYCLIZATION ZAMBON S.P.A. (IT) 1988-09-20 US disclosed
EP-0207955-A1 PROCESS FOR THE PREPARATION OF 3,5-DISUBSTITUTED ISOXAZOLES. ZAMBON SPA (IT) 1987-01-14 EP disclosed
WO-1986003490-A1 PROCESS FOR THE PREPARATION OF 3,5-DISUBSTITUTED ISOXAZOLES ZAMBON S.P.A. (IT) 1986-06-19 WO disclosed