SCHEMBL8882015

SCHEMBL8882015

CC(C)C(S)C(=O)NC1=CCc2ccc(-c3ccccc3)cc2N(CC(=O)O)C1=O

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACE P12821 9/20 0.39
MME P08473 8/20 0.39
CPA1 P15085 2/20 0.39
ACE2 Q9BYF1 2/20 0.39
XIAP P98170 2/20 0.34
AKR1B1 P15121 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
ECE1 P42892 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8881495 0.86 MME (0.45) ACEMMECPA1ACE2
SCHEMBL9227091 0.73 ACE (0.56) ACEMME
SCHEMBL8883149 0.73 ACE (0.56) ACEMME
SCHEMBL8882317 0.72 MMEL1 (0.36)
SCHEMBL8881756 0.68 ALDH1A1 (0.36)
SCHEMBL14865944 0.60 BRD4 (0.47)
SCHEMBL11109826 0.55 CA12 (0.44) CA12CA9
SCHEMBL8673301 0.55 ALDH1A1 (0.48) HDAC1HDAC6
SCHEMBL522099 0.55 ALDH1A1 (0.50) CA12CA9
SCHEMBL24879174 0.55 TAAR1 (0.70) ACEMMECPA1ACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5679671-A ANGIOTENSIN 1-CONVERTING ENZYME INHIBITOR, VASOPRESSIN ANTAGONISM AND ATRIAL NAUTRIURETIC PEPTIDE HYDROLASE INHIBITOR EISAI CO., LTD. (JP) 1997-10-21 US disclosed