SCHEMBL8882974

SCHEMBL8882974

O=C1CC(C(=O)O)(C(=O)O)CN1Cc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.46
POLB P06746 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.46
DDB1 Q16531 1/20 0.44
CRBN Q96SW2 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
RIPK1 Q13546 1/20 0.44
HDAC6 Q9UBN7 1/20 0.43
MEN1 O00255 1/20 0.43
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
GAA P10253 2/20 0.41
EPHX2 P34913 1/20 0.41
GRM6 O15303 1/20 0.40
BRD4 O60885 1/20 0.40
ALDH1A1 P00352 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8881749 0.86 NPSR1 (0.43) KMT2APOLBCYP2D6CYP2C9CYP2C19
SCHEMBL8882202 0.85 CASP3 (0.46) KMT2APOLBCYP2D6CYP2C9CYP2C19
SCHEMBL9233093 0.84 L3MBTL1 (0.49) KMT2APOLBCYP2D6CYP2C9CYP2C19
SCHEMBL8881736 0.82 CASP3 (0.46) KMT2APOLBCYP2D6CYP2C9CYP2C19
SCHEMBL26965325 0.77 RIPK1 (0.44) KMT2APOLBCYP2D6CYP2C9CYP2C19
SCHEMBL17925766 0.77 GAA (0.51) KMT2APOLBCYP2D6CYP2C9CYP2C19
SCHEMBL9233372 0.76 KDM4E (0.41) KMT2APOLBCYP2D6CYP2C9CYP2C19
SCHEMBL8881539 0.75 NPSR1 (0.41) KMT2APOLBCYP2D6CYP2C9CYP2C19
SCHEMBL8881874 0.74 RAB9A (0.40) KMT2ACYP2D6CYP2C9CYP2C19L3MBTL1
SCHEMBL8882513 0.74 CASP3 (0.47) KMT2ACYP2D6CYP2C9CYP2C19PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5677316-A BACTERICIDES YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-10-14 US disclosed
EP-0677522-A1 8-METHOXYQUINOLONECARBOXYLIC ACID DERIVATIVE YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-10-18 EP disclosed