SCHEMBL8883136

SCHEMBL8883136

O=C(O)c1ncccc1OCc1ccc(Cl)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPIA P62937 4/20 0.55
HPGD P15428 1/20 0.51
RXRA P19793 1/20 0.51
RXRB P28702 1/20 0.51
L3MBTL1 Q9Y468 4/20 0.51
NR4A2 P43354 2/20 0.50
MRGPRX4 Q96LA9 2/20 0.49
LMNA P02545 1/20 0.47
GAA P10253 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
RHEB Q15382 1/20 0.46
MAPK1 P28482 1/20 0.46
MEN1 O00255 1/20 0.46
NPC1 O15118 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
MAPT P10636 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2426791 0.88 LTA4H (0.58) PPIAHPGDRXRARXRBLTA4H
SCHEMBL30848623 0.88 LTA4H (0.58) PPIAHPGDRXRARXRBLTA4H
SCHEMBL8883987 0.87 KMT2A (0.56) PPIAHPGDRXRARXRBL3MBTL1
Hydrochloric Acid SCHEMBL10705444 0.86 LTA4H (0.57) PPIAHPGDRXRARXRBLTA4H
SCHEMBL8883336 0.86 L3MBTL1 (0.63) PPIAL3MBTL1MRGPRX4LMNAGAA
SCHEMBL8883654 0.85 RXRA (0.50) PPIAHPGDRXRARXRBL3MBTL1
SCHEMBL8883647 0.85 ABCB1 (0.50) PPIAHPGDRXRARXRBL3MBTL1
SCHEMBL8881868 0.85 RXRA (0.53) PPIAHPGDRXRARXRBL3MBTL1
SCHEMBL8882076 0.85 RXRA (0.56) PPIAHPGDRXRARXRBNR4A2
SCHEMBL8883184 0.85 NPC1 (0.63) HPGDRXRARXRBMRGPRX4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658933-A Substituted heterocyclic carboxamide esters, their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-08-19 US disclosed
CN-1107145-A Substituted heterocyclic carboxamides, their preparation and their use as pharmaceuticals HOECHST AG (DE) 1995-08-23 CN disclosed
CN-1107144-A Substituted heterocyclic carboxamide esters, their preparation and their use as pharmaceuticals HOECHST AG (DE) 1995-08-23 CN disclosed
EP-0650961-A1 Substituted heterocyclic carboxylic acid amides, their preparation, and their use as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-05-03 EP disclosed
EP-0650960-A1 Substituted heterocyclic carboxylic acid amide esters, their preparation and their us as medicaments HOECHST AKTIENGESELLSCHAFT (DE) 1995-05-03 EP disclosed