SCHEMBL8883709

SCHEMBL8883709

CCOc1nc(NC(C)=O)nc2c1NC=[N+]2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 2/20 0.37
PRKD3 O94806 1/20 0.37
MAP4K4 O95819 1/20 0.37
MAPK9 P45984 1/20 0.37
MAPK10 P53779 1/20 0.37
MAP4K2 Q12851 1/20 0.37
PKN2 Q16513 1/20 0.37
PRKD2 Q9BZL6 1/20 0.37
STK17A Q9UEE5 1/20 0.37
CYP1A2 P05177 2/20 0.36
TDP1 Q9NUW8 2/20 0.35
MEN1 O00255 1/20 0.35
LMNA P02545 1/20 0.35
KMT2A Q03164 1/20 0.35
ALDH1A1 P00352 2/20 0.35
MAPT P10636 1/20 0.33
ADORA3 P0DMS8 4/20 0.33
KDM4E B2RXH2 1/20 0.33
ALPL P05186 1/20 0.33
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8781884 0.78 CYP1A2 (0.38) CYP1A2KMT2AALDH1A1MAPTADORA3
SCHEMBL8886489 0.70 HTR1A (0.35) CYP1A2TDP1LMNAADORA3KDM4E
SCHEMBL9640561 0.67 CYP1A2 (0.66) MAPK8PRKD3MAP4K4MAPK9MAPK10
SCHEMBL9564706 0.66 ALDH1A1 (0.31) ALDH1A1
SCHEMBL8883705 0.66 MAPK8 (0.39) MAPK8PRKD3MAP4K4MAPK9MAPK10
SCHEMBL536840 0.65 L3MBTL1 (0.40) MEN1LMNAKMT2AALDH1A1MAPT
SCHEMBL19186680 0.65 CDK1 (0.41) MAPK8PRKD3MAP4K4MAPK9MAPK10
SCHEMBL4119354 0.64 MAPK8 (0.40) MAPK8PRKD3MAP4K4MAPK9MAPK10
SCHEMBL15781042 0.62 CDK5 (0.49) TDP1MAPTKDM4E
SCHEMBL3331750 0.61 TTK (0.48) MAPK8MAPK10CYP1A2TDP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5631259-A PURINE BASE DERIVATIVES FOR NUCLEOSIDES HOECHST AKTIENGESELLSCHAFT (DE) 1997-05-20 US claimed
US-5631259-A PURINE BASE DERIVATIVES FOR NUCLEOSIDES HOECHST AKTIENGESELLSCHAFT (DE) 1997-05-20 US disclosed
EP-0521463-A2 Substituted cyclic cycloalkyltriols, process, intermediates for their preparation and their use as antiviral and antiparasitic agents HOECHST AKTIENGESELLSCHAFT (DE) 1993-01-07 EP disclosed