SCHEMBL8885671

SCHEMBL8885671

O=CC1=C(O)c2ccccc2CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.47
MIF P14174 5/20 0.41
ESR1 P03372 1/20 0.40
SRD5A1 P18405 1/20 0.40
SRD5A2 P31213 1/20 0.40
MAOB P27338 2/20 0.39
CYP2A6 P11509 1/20 0.38
MAOA P21397 1/20 0.38
RAB9A P51151 3/20 0.37
ALDH1A1 P00352 2/20 0.37
NPC1 O15118 2/20 0.37
MAPT P10636 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MITF O75030 1/20 0.37
HSP90AA1 P07900 1/20 0.37
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
KDM4E B2RXH2 2/20 0.37
LMNA P02545 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29952458 0.81 ESR1 (0.54) CES1ESR1SRD5A1SRD5A2MAOB
SCHEMBL2063760 0.81 ESR1 (0.54) CES1ESR1SRD5A1SRD5A2MAOB
SCHEMBL29615759 0.77 CES1 (0.47) CES1MIFESR1SRD5A1SRD5A2
SCHEMBL4268656 0.77 CES1 (0.47) CES1MIFESR1SRD5A1SRD5A2
SCHEMBL16139564 0.74 CES1 (0.44) CES1MIFSRD5A1SRD5A2MAOB
SCHEMBL4271075 0.73 LMNA (0.42) CES1ESR1SRD5A1SRD5A2MAOB
SCHEMBL12797026 0.70 ESR1 (0.56) CES1MIFESR1MAOBCYP2A6
SCHEMBL19645160 0.69 CES1 (0.46) CES1MIFSRD5A1SRD5A2MAOB
SCHEMBL24282949 0.69 ALDH1A1 (0.51) CES1SRD5A1SRD5A2MAOBCYP2A6
SCHEMBL24512062 0.69 CES1 (0.35) CES1MIFESR1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5670522-A Dopamine receptor subtype ligands MERCK SHARP & DOHME LIMITED (GB) 1997-09-23 US disclosed
US-5670522-A Dopamine receptor subtype ligands MERCK SHARP & DOHME LIMITED (GB) 1997-09-23 US disclosed
EP-0665840-A1 DOPAMINE RECEPTOR SUBTYPE LIGANDS MERCK SHARP & DOHME LTD. (GB) 1995-08-09 EP disclosed
EP-0665840-A1 DOPAMINE RECEPTOR SUBTYPE LIGANDS MERCK SHARP & DOHME LTD. (GB) 1995-08-09 EP disclosed
WO-1994010162-A1 DOPAMINE RECEPTOR SUBTYPE LIGANDS MERCK SHARP & DOHME LIMITED (GB) 1994-05-11 WO disclosed
WO-1994010162-A1 DOPAMINE RECEPTOR SUBTYPE LIGANDS MERCK SHARP & DOHME LIMITED (GB) 1994-05-11 WO disclosed