SCHEMBL8886474

SCHEMBL8886474

Cc1ccc(C(N)=Nc2ccc(S(C)(=O)=O)cc2)nc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.40
ADRA2A P08913 2/20 0.40
ADRA2B P18089 2/20 0.40
ADRA2C P18825 2/20 0.40
PLAU P00749 2/20 0.40
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
GPR119 Q8TDV5 1/20 0.38
HTR3E A5X5Y0 1/20 0.38
SLC22A2 O15244 1/20 0.38
SLC22A1 O15245 1/20 0.38
SLC22A3 O75751 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
F2 P00734 2/20 0.36
PRSS1 P07477 2/20 0.36
PRSS2 P07478 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5594310 0.80 PLAU (0.41) PTGS2PLAUNOS3NOS1NOS2
SCHEMBL5594064 0.79 KDM4E (0.50) PTGS2NOS3NOS1NOS2PTGS1
SCHEMBL4854998 0.78 CYP2D6 (0.60) PTGS2PLAUNOS3NOS1NOS2
SCHEMBL5595201 0.78 CYP2D6 (0.60) PTGS2PLAUNOS3NOS1NOS2
SCHEMBL5594294 0.78 P2RX7 (0.41) PTGS2NOS3NOS1NOS2PTGS1
SCHEMBL5594531 0.77 NOS3 (0.51) ADRA2AADRA2BADRA2CPLAUNOS3
SCHEMBL5594283 0.75 ADRA2A (0.46) PTGS2ADRA2AADRA2BADRA2CNOS3
SCHEMBL7451804 0.74 PTGS2 (0.45) PTGS2GPR119
SCHEMBL5594753 0.72 P2RX7 (0.43) PTGS2PLAUNOS3NOS1NOS2
SCHEMBL11879362 0.71 POLB (0.58) ADRA2AADRA2BADRA2CPLAUNOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5616601-A 1,2-aryl and heteroaryl substituted imidazolyl compounds for the treatment of inflammation GD SEARLE & CO (US) 1997-04-01 US disclosed