SCHEMBL8889779

SCHEMBL8889779

COc1ccc(C(=O)Nc2c(Cl)cncc2Cl)cc1COc1ccccn1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 11/20 0.61
PDE4B Q07343 11/20 0.57
PDE4A P27815 8/20 0.57
PDE4C Q08493 8/20 0.57
CYP2B6 P20813 1/20 0.56
KMT2A Q03164 2/20 0.51
MAPK1 P28482 1/20 0.51
HDAC8 Q9BY41 1/20 0.46
SGMS2 Q8NHU3 1/20 0.46
POLB P06746 1/20 0.45
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
ABCB11 O95342 1/20 0.44
GRM4 Q14833 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8888978 0.87 PDE4D (0.65) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8890145 0.84 PDE4D (0.61) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8889907 0.82 PDE4D (0.64) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8888975 0.82 PDE4D (0.70) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8892872 0.80 KMT2A (0.55) KMT2AMAPK1MEN1ALDH1A1CYP1A2
SCHEMBL8891532 0.80 PDE4D (0.66) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8891152 0.79 PDE4D (0.62) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8890162 0.79 KMT2A (0.53) KMT2AMAPK1MEN1ALDH1A1
SCHEMBL8891655 0.78 PDE4B (0.70) PDE4DPDE4BPDE4APDE4CCYP2B6
SCHEMBL8889614 0.78 PDE4D (0.73) PDE4DPDE4BPDE4APDE4CCYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO claimed
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO disclosed