SCHEMBL8890166

SCHEMBL8890166

COCCNc1nc(NCCCCCC(N)=O)nc2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.52
CYP1A2 P05177 8/20 0.51
CYP3A4 P08684 8/20 0.51
USP2 O75604 4/20 0.51
ALOX15 P16050 3/20 0.51
CLK4 Q9HAZ1 3/20 0.51
ALDH1A1 P00352 3/20 0.51
TP53 P04637 2/20 0.51
APEX1 P27695 1/20 0.51
CASP7 P55210 1/20 0.51
HSD17B10 Q99714 4/20 0.49
ACHE P22303 3/20 0.49
APP P05067 2/20 0.49
KDM4E B2RXH2 2/20 0.49
CASP6 P55212 1/20 0.49
CYP2D6 P10635 3/20 0.48
CYP2C19 P33261 3/20 0.48
TSHR P16473 3/20 0.48
MAPK1 P28482 1/20 0.48
SIRT5 Q9NXA8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8890175 0.86 PDE5A (0.55) PDE5ACYP1A2CYP3A4USP2ALOX15
SCHEMBL8890389 0.85 ACHE (0.48) ACHEAPPCASP6SIRT5RAD52
Hydrochloric Acid SCHEMBL8890506 0.82 POLB (0.59) ACHEAPPCASP6SIRT5
SCHEMBL8892539 0.79 NPY5R (0.60) ALOX15TP53APPTSHRMAPK1
SCHEMBL6039576 0.79 NPY5R (0.60) ALOX15TP53APPTSHRMAPK1
SCHEMBL8891176 0.79 NPY5R (0.60) ALOX15TP53APPTSHRMAPK1
Hydrochloric Acid SCHEMBL8892580 0.78 NPY5R (0.58) ALOX15ALDH1A1TP53APPKDM4E
SCHEMBL8893012 0.77 ADRA2A (0.47)
SCHEMBL8898351 0.76 VCP (0.48) PDE5ACYP1A2CYP3A4USP2ALOX15
SCHEMBL8889077 0.75 VCP (0.47) ACHEAPPCASP6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020821-A1 HETEROARYL DERIVATIVES NOVARTIS AG (CH) 1997-06-12 WO disclosed