SCHEMBL8890175

SCHEMBL8890175

COCCNc1nc(NCCCCCCN)nc2ccccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.55
CASP6 P55212 1/20 0.53
CYP1A2 P05177 9/20 0.53
CYP3A4 P08684 9/20 0.53
HSD17B10 Q99714 4/20 0.53
KDM4E B2RXH2 2/20 0.53
CYP2C19 P33261 4/20 0.52
CYP2D6 P10635 4/20 0.52
USP2 O75604 4/20 0.52
CLK4 Q9HAZ1 3/20 0.52
ALOX15 P16050 2/20 0.52
ALDH1A1 P00352 2/20 0.52
MAPK1 P28482 1/20 0.52
TSHR P16473 4/20 0.52
LDHA P00338 1/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
APP P05067 2/20 0.50
BCHE P06276 2/20 0.50
ACHE P22303 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8890166 0.86 PDE5A (0.52) PDE5ACASP6CYP1A2CYP3A4HSD17B10
SCHEMBL11734758 0.85 CASP6 (0.62) CASP6KDM4EALDH1A1KMT2AAPP
SCHEMBL8890399 0.84 CASP6 (0.52) CASP6APPBCHEACHERAD52
SCHEMBL8890767 0.81 POLB (0.61) CASP6ALDH1A1MAPK1APPBCHE
Hydrochloric Acid SCHEMBL8890527 0.81 POLB (0.64) CASP6ALDH1A1MAPK1APPBCHE
SCHEMBL8898526 0.77 CYP1A2 (0.50) PDE5ACASP6CYP1A2CYP3A4HSD17B10
SCHEMBL8893524 0.77 NPY5R (0.70) ALOX15MAPK1TSHRAPPACHE
SCHEMBL4779679 0.77 APP (0.71) CYP1A2CYP3A4HSD17B10KDM4ECYP2C19
SCHEMBL8892545 0.77 NPY5R (0.70) ALOX15MAPK1TSHRAPPACHE
SCHEMBL6039582 0.77 NPY5R (0.70) ALOX15MAPK1TSHRAPPACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020821-A1 HETEROARYL DERIVATIVES NOVARTIS AG (CH) 1997-06-12 WO disclosed