SCHEMBL8890233

SCHEMBL8890233

O=C1Nc2cc(OCc3ccccc3)ccc2Nc2ccccc21

nearest known ligand 0.69

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAOA P21397 11/20 0.69
MAOB P27338 11/20 0.69
TNKS2 Q9H2K2 2/20 0.54
PDGFRA P16234 1/20 0.54
FER P16591 1/20 0.54
LTK P29376 1/20 0.54
CDK8 P49336 1/20 0.54
ACVR1 Q04771 1/20 0.54
LRRK2 Q5S007 1/20 0.54
DYRK1B Q9Y463 1/20 0.54
CSNK1G1 Q9HCP0 1/20 0.54
CHEK1 O14757 1/20 0.54
CREBBP Q92793 1/20 0.53
TOP1 P11387 1/20 0.49
GSTP1 P09211 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9728150 0.82 MAOB (1.00) MAOAMAOBTOP1GSTP1
SCHEMBL9183428 0.80 EDNRA (0.60) MAOAMAOBPDGFRAFERLTK
SCHEMBL27634033 0.79 MAOA (1.00) MAOAMAOBTOP1GSTP1
SCHEMBL26547707 0.77 MAOB (0.55) MAOAMAOBCREBBPTOP1
SCHEMBL7379163 0.77 MAOA (1.00) MAOAMAOBTOP1GSTP1
SCHEMBL20520341 0.76 MAOA (0.79) MAOAMAOBCREBBPTOP1GSTP1
SCHEMBL30536411 0.75 CES1 (0.62) PDGFRAFERLTKCDK8ACVR1
SCHEMBL9179367 0.74 MAOB (0.47) MAOAMAOBTNKS2CREBBP
SCHEMBL6351678 0.74 MAOA (0.62) MAOAMAOBTNKS2CREBBPTOP1
SCHEMBL6351677 0.74 MAOA (0.62) MAOAMAOBTNKS2CREBBPTOP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997000252-A1 TRICYCLIC INHIBITORS OF PROTEIN FARNESYLTRANSFERASE WARNER-LAMBERT COMPANY (US) 1997-01-03 WO disclosed
US-5420123-A Dibenzodiazepine endothelin antagonists BRISTOL-MYERS SQUIBB COMPANY (US) 1995-05-30 US disclosed