SCHEMBL8891429

SCHEMBL8891429

CN(C)Cc1cccc2c(Nc3ccccc3)nc(Nc3ccc(CS(=O)(=O)N(C)C)cc3)nc12

nearest known ligand 0.72

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 9/20 0.72
PDE5A O76074 1/20 0.39
EGFR P00533 1/20 0.38
ITK Q08881 1/20 0.38
KDM1A O60341 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
HSD17B10 Q99714 1/20 0.38
NEK2 P51955 1/20 0.37
CCNT1 O60563 1/20 0.37
CCNE1 P24864 1/20 0.37
CDK2 P24941 1/20 0.37
CDK9 P50750 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8899629 0.99 NPY5R (0.71) NPY5RPDE5AEGFRITKKDM1A
SCHEMBL8891585 0.87 NPY5R (0.77) NPY5RPDE5AEGFRITKKDM1A
Hydrochloric Acid SCHEMBL8890940 0.86 NPY5R (0.75) NPY5RPDE5AEGFRITKKDM1A
SCHEMBL8890967 0.85 NPY5R (0.74) NPY5RKDM1A
SCHEMBL8898853 0.84 NPY5R (1.00) NPY5RPDE5A
Hydrochloric Acid SCHEMBL8900310 0.84 NPY5R (0.72) NPY5RKDM1A
Hydrochloric Acid SCHEMBL8900633 0.83 NPY5R (0.98) NPY5RPDE5A
SCHEMBL8891909 0.78 NPY5R (0.83) NPY5RPDE5AEGFR
SCHEMBL8889462 0.77 NPY5R (0.62) NPY5RKDM1ANEK2
SCHEMBL8900516 0.77 NPY5R (0.77) NPY5RALDH1A1CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020822-A1 QUINAZOLIN-2,4-DIAZIRINES AS NPY RECEPTOR ANTAGONIST NOVARTIS AG (CH) 1997-06-12 WO claimed