SCHEMBL8891722

SCHEMBL8891722

N=CSCc1ccc(N2CC(C(=O)N3CCN(CC(=O)OCc4ccccc4)CC3)OC2=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
HPGD P15428 1/20 0.34
GRM2 Q14416 1/20 0.34
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34
AVPR1A P37288 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
PREP P48147 1/20 0.33
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33
TMEM97 Q5BJF2 2/20 0.33
SIGMAR1 Q99720 2/20 0.33
ADRB1 P08588 1/20 0.33
HRH1 P35367 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8891141 0.87 ITGB3 (0.40) ITGB3ITGA2BHPGDGRM2CA1
SCHEMBL8892077 0.85 ITGB3 (0.43) ITGB3ITGA2BHPGD
SCHEMBL8894919 0.84 ITGB3 (0.40) ITGB3ITGA2BHPGDGRM2PPARG
SCHEMBL8891751 0.84 FNTA (0.45) ITGB3ITGA2BGRM2POLBHRH1
SCHEMBL8893028 0.83 ITGB3 (0.43) ITGB3ITGA2BHPGDGRM2CA1
SCHEMBL8892340 0.80 MEN1 (0.42) ITGB3ITGA2BCA1CA2CA7
SCHEMBL8894032 0.79 ITGB3 (0.45) ITGB3ITGA2B
SCHEMBL7457368 0.77 ITGB3 (0.41) ITGB3ITGA2BTMEM97SIGMAR1HRH1
SCHEMBL8891713 0.75 KMT2A (0.32) ITGB3ITGA2BHPGDPPARGPPARA
SCHEMBL8892670 0.74 NPC1 (0.40) ITGB3HPGDCA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5614535-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-03-25 US disclosed