SCHEMBL8892597

SCHEMBL8892597

COC(=O)Cn1c(=O)[nH]c(=O)c2c(Cl)cc(Cl)cc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CBX7 O95931 1/20 0.42
CDYL2 Q8N8U2 1/20 0.42
CDYL Q9Y232 1/20 0.42
CDY1; CDY1B Q9Y6F8 1/20 0.42
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
MEN1 O00255 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KAT2B Q92831 1/20 0.38
CHEK1 O14757 1/20 0.38
WEE1 P30291 1/20 0.38
ALDH1A1 P00352 2/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10487991 0.88 ALDH1A1 (0.46) KDM4ESMN1; SMN2MEN1CYP3A4CYP2C9
SCHEMBL8890391 0.85 HDAC6 (0.58) KDM4ESMN1; SMN2CBX7CDYL2CDYL
SCHEMBL8893031 0.84 GRIN2D (0.48) CBX7CDYL2CDYLCDY1; CDY1BHDAC1
SCHEMBL8432918 0.80 CBX7 (0.47) KDM4ESMN1; SMN2CBX7CDYL2CDYL
SCHEMBL8901340 0.77 KDM4E (0.40) KDM4ESMN1; SMN2HDAC1HDAC8HDAC6
Hydrochloric Acid SCHEMBL8890311 0.75 ITGB1 (0.37) KDM4EHDAC1HDAC8HDAC6ALDH1A1
SCHEMBL8487616 0.73 KDM4E (0.59) KDM4ESMN1; SMN2MEN1CYP3A4CYP2C9
SCHEMBL10488076 0.72 HDAC1 (0.53) KDM4EHDAC1HDAC8HDAC6MEN1
SCHEMBL7231747 0.70 KDM4E (0.67) KDM4ESMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL8907357 0.68 CA12 (0.38) MEN1CYP2C9CYP2C19KMT2AGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997002254-A1 QUINAZOLINE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-01-23 WO disclosed