SCHEMBL8892927

SCHEMBL8892927

CN(C1CCCCC1)C1(C(N)=O)CCN(Cc2ccccc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.55
CYP2D6 P10635 2/20 0.53
ALDH1A1 P00352 1/20 0.53
CHRM2 P08172 4/20 0.46
CHRM3 P20309 4/20 0.46
HRH3 Q9Y5N1 1/20 0.46
ACHE P22303 3/20 0.46
SIGMAR1 Q99720 2/20 0.45
DRD2 P14416 1/20 0.45
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
HTR2B P41595 1/20 0.45
OPRM1 P35372 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5127015 0.84 CYP2D6 (0.60) TSHRCYP2D6ALDH1A1CHRM2CHRM3
SCHEMBL8894213 0.76 OPRM1 (0.50) CHRM2CHRM3HRH3ACHESIGMAR1
SCHEMBL11889046 0.76 CYP2D6 (0.58) TSHRCYP2D6ALDH1A1CHRM2CHRM3
SCHEMBL12861220 0.74 CYP2D6 (0.61) TSHRCYP2D6ALDH1A1CHRM2CHRM3
SCHEMBL16876722 0.74 TSHR (0.54) TSHRCYP2D6ALDH1A1CHRM2CHRM3
SCHEMBL14716240 0.73 CYP2D6 (0.63) TSHRCYP2D6ALDH1A1CHRM2CHRM3
SCHEMBL23647380 0.72 TSHR (0.58) TSHRCYP2D6ALDH1A1CHRM2CHRM3
SCHEMBL27473621 0.72 SIGMAR1 (0.65) CHRM2CHRM3ACHESIGMAR1DRD2
SCHEMBL8892930 0.72 ALDH1A1 (0.62) TSHRCYP2D6ALDH1A1HRH3OPRM1
SCHEMBL7313593 0.71 CACNA1G (0.53) TSHRCYP2D6ALDH1A1CHRM2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5610142-A Bradykinin antagonist pseudopeptide derivatives of substituted 4-keto-1,3,8-triazaspiro[4.5]decan-3-alkanoic acids SCIOS INC. (US) 1997-03-11 US disclosed