SCHEMBL8893433

SCHEMBL8893433

Fc1ccccc1C(OCCN1CCC1)c1ccccc1F

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.55
SIGMAR1 Q99720 4/20 0.51
SLC6A4 P31645 4/20 0.49
SLC6A3 Q01959 4/20 0.49
CYP3A4 P08684 3/20 0.49
SLC6A2 P23975 3/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 2/20 0.49
TSHR P16473 2/20 0.49
CYP2C19 P33261 2/20 0.49
HIF1A Q16665 2/20 0.49
KCNH2 Q12809 2/20 0.49
SLC22A1 O15245 1/20 0.49
CHRM2 P08172 1/20 0.49
HTR1A P08908 1/20 0.49
ADRA2A P08913 1/20 0.49
CHRM1 P11229 1/20 0.49
DRD1 P21728 1/20 0.49
TBXA2R P21731 1/20 0.49
ADRA1A P35348 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8892312 0.97 CHRNA7 (0.58) CHRNA7SIGMAR1SLC6A4SLC6A3CYP3A4
SCHEMBL8892798 0.95 CHRNA7 (0.60) CHRNA7SIGMAR1SLC6A4SLC6A3CYP3A4
SCHEMBL11073631 0.80 SLC6A4 (0.74) SLC6A4SLC6A3SLC6A2
SCHEMBL8642037 0.74 LMNA (0.78) SIGMAR1SLC6A4SLC6A3CYP3A4SLC6A2
SCHEMBL8893211 0.74 IDO1 (0.35) CHRNA7SIGMAR1SLC6A4SLC6A3CYP3A4
Perastine SCHEMBL1506306 0.72 CYP3A4 (0.83) CHRNA7SIGMAR1SLC6A4SLC6A3CYP3A4
SCHEMBL7423150 0.72 CHRNA7 (0.65) CHRNA7SIGMAR1SLC6A4SLC6A3CYP3A4
SCHEMBL8647649 0.71 LMNA (0.83) SIGMAR1SLC6A4SLC6A3CYP3A4SLC6A2
Perastine SCHEMBL29768269 0.71 CYP3A4 (0.83) CHRNA7SIGMAR1SLC6A4SLC6A3CYP3A4
SCHEMBL10357800 0.71 SIGMAR1 (0.81) SIGMAR1SLC6A4SLC6A3CYP3A4SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997027175-A1 SUBSTITUTED ETHYL α,α - DIARYLMETHYL ETHER DERIVATIVES GUILFORD PHARMACEUTICALS INC. (US) 1997-07-31 WO claimed