SCHEMBL8894440

SCHEMBL8894440

CCC(=O)c1cc(Cl)c(C)cc1OC

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 1/20 0.51
GAA P10253 1/20 0.44
TSHR P16473 3/20 0.43
GLA P06280 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.41
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
RAB9A P51151 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HTR4 Q13639 7/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
HTR3A P46098 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9720549 0.87 HMGCR (0.51) HMGCRGAATSHRSMN1; SMN2ALDH1A1
SCHEMBL8895935 0.86 HMGCR (0.54) HMGCRGAATSHRSMN1; SMN2ALDH1A1
SCHEMBL9720676 0.86 HMGCR (0.58) HMGCRKDM4EALDH1A1CYP3A4KMT2A
SCHEMBL23174248 0.85 GAA (0.43) GAATSHRGLASMN1; SMN2KDM4E
SCHEMBL2099536 0.85 HPGDS (0.45) GAATSHRGLASMN1; SMN2KDM4E
SCHEMBL11342543 0.84 HMGCR (0.61) HMGCRGAAALDH1A1CYP3A4KMT2A
SCHEMBL11807436 0.81 GAA (0.47) GAATSHRGLASMN1; SMN2KDM4E
SCHEMBL3928834 0.81 GAA (0.47) GAATSHRGLASMN1; SMN2KDM4E
SCHEMBL7802404 0.81 ALDH1A1 (0.51) GAATSHRGLASMN1; SMN2KDM4E
SCHEMBL5643886 0.80 HMGCR (0.51) HMGCRTSHRSMN1; SMN2KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5656648-A TREATMENT OF PATHOLOGIES NECESSITATING STIMULATION OF CHOLECYSTOKININ-A RECEPTORS BY TOTAL OR PARTIAL AGONIST EFFECT SANOFI (FR) 1997-08-12 US disclosed
EP-0611766-A1 Polysubstituted 2-amido thiazoles derivatives, process for their preparation, pharmaceutical compositions and utilization for the preparation of a medicament SANOFI (FR) 1994-08-24 EP disclosed
US-5103022-A Reacting dl-2-methyl-1-(4-trifluoromethylphenyl)-3-pyrrolidino -1-propanone with l-acetylphenylglycine to form corresponding diastereomeric salt, deposition, isolation of l-2-methyl-1-(4-trifluoromethylphenyl)-3-pyrrolidino-1-propanone NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1992-04-07 US disclosed
US-5057535-A Muscle relaxants NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1991-10-15 US disclosed
EP-0200942-A2 New derivatives of an aminoketone NIPPON KAYAKU KABUSHIKI KAISHA (JP) 1986-11-12 EP disclosed