SCHEMBL8905206

SCHEMBL8905206

CC(=O)NS(=O)(=O)n1cc(C(F)(F)F)nc1-c1cc(C)cc(Cl)c1

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 19/20 0.53
PTGS1 P23219 9/20 0.39
SYK P43405 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8896836 0.83 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL5069835 0.79 PTGS2 (0.73) PTGS2PTGS1
SCHEMBL8894968 0.73 PTGS2 (0.55) PTGS2PTGS1
SCHEMBL8343845 0.71 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL8347213 0.70 PTGS2 (0.55) PTGS2PTGS1SYK
SCHEMBL5594003 0.70 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL5069832 0.69 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL8923114 0.67 PTGS2 (0.62) PTGS2PTGS1
SCHEMBL8347217 0.67 PTGS2 (0.69) PTGS2PTGS1
SCHEMBL12258055 0.64 PKM (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997038986-A1 SUBSTITUTED BENZENESULFONAMIDE DERIVATIVES AS PRODRUGS OF COX-2 INHIBITORS G.D. SEARLE & CO. (US) 1997-10-23 WO disclosed