SCHEMBL8899666

SCHEMBL8899666

CC(=O)N(I)C(C)Nc1ccc2ccccc2c1S(=O)(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCEH1 Q6PIU2 3/20 0.36
CYP2D6 P10635 1/20 0.36
METAP2 P50579 2/20 0.34
METAP1 P53582 1/20 0.34
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
CA12 O43570 1/20 0.33
CA4 P22748 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
MAPT P10636 2/20 0.33
HPGD P15428 2/20 0.33
KEAP1 Q14145 1/20 0.32
HSD17B10 Q99714 1/20 0.32
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18268231 0.80 IDO1 (0.46) NCEH1CYP2D6METAP2METAP1KDM4E
SCHEMBL2524191 0.78 CYP2D6 (0.38) CYP2D6METAP2METAP1KDM4ECA12
SCHEMBL3765915 0.76 ANPEP (0.36) NCEH1CYP2D6METAP2METAP1ALDH1A1
SCHEMBL8928010 0.76 ANPEP (0.36) NCEH1CYP2D6METAP2METAP1ALDH1A1
SCHEMBL590579 0.75 CYP1A2 (0.43) CYP1A2CA9CASP6
SCHEMBL5173798 0.74 ALDH1A1 (0.54) CYP2D6METAP2METAP1ALDH1A1KDM4E
SCHEMBL6335916 0.74 CYP2D6 (0.44) CYP2D6METAP2METAP1ALDH1A1KDM4E
SCHEMBL5699450 0.72 IDO1 (0.46) CYP2D6METAP2METAP1ALDH1A1KEAP1
SCHEMBL2951963 0.72 CYP2D6 (0.39) CYP2D6METAP2METAP1ALDH1A1KDM4E
SCHEMBL6032490 0.71 SLC2A1 (0.36) CYP2D6METAP2METAP1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0758681-A2 Inhibiting transformation of cells having elevated purine metabolic enzyme activity MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1997-02-19 EP disclosed
EP-0458901-A1 INHIBITING TRANSFORMATION OF CELLS HAVING ELEVATED PURINE METABOLIC ENZYME ACTIVITY MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1991-12-04 EP disclosed
WO-1990009192-A1 INHIBITING TRANSFORMATION OF CELLS HAVING ELEVATED PURINE METABOLIC ENZYME ACTIVITY MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1990-08-23 WO disclosed