SCHEMBL8899787

SCHEMBL8899787

CC(C)(C)OC(=O)N1CCC(CNS(=O)(=O)c2cccc3ccccc23)CC1

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 16/20 0.64
KDM4E B2RXH2 2/20 0.56
PKM P14618 1/20 0.56
NPY5R Q15761 2/20 0.55
NPY1R P25929 1/20 0.55
MAPT P10636 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8890529 0.91 TGFBR1 (0.53) TGFBR1KDM4EPKMNPY5R
SCHEMBL27917809 0.85 NPY5R (0.58) NPY5RNPY1RMAPT
SCHEMBL14834135 0.84 MGLL (0.64) TGFBR1NPY5RNPY1RMAPT
SCHEMBL14695860 0.84 TGFBR1 (0.79) TGFBR1KDM4EPKM
SCHEMBL6039411 0.83 ACACB (0.69) NPY5RNPY1RMAPT
SCHEMBL6039406 0.83 ACACB (0.69) NPY5RNPY1RMAPT
SCHEMBL10194489 0.82 ACACB (0.71) TGFBR1
SCHEMBL8899558 0.81 ACKR3 (0.53) NPY5RNPY1R
SCHEMBL8899052 0.79 NPY5R (0.55) TGFBR1NPY5RNPY1RMAPT
SCHEMBL8899046 0.79 NPY5R (0.55) TGFBR1NPY5RNPY1RMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020820-A1 HETEROARYL COMPOUNDS NOVARTIS AG (CH) 1997-06-12 WO disclosed